SCHEMBL5201900

SCHEMBL5201900

Cc1nnc(C(=O)NCC(C)c2nc(C(=O)N(C)Cc3ccc(F)cc3)c(O)c(=O)[nH]2)o1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.43
THRB P10828 2/20 0.43
TP53 P04637 1/20 0.43
KCNE1 P15382 1/20 0.42
CCR1 P32246 1/20 0.42
KCNQ1 P51787 1/20 0.42
ERCC1 P07992 2/20 0.38
FEN1 P39748 2/20 0.38
ERCC4 Q92889 2/20 0.38
RAB9A P51151 1/20 0.37
LIPE Q05469 1/20 0.34
ELANE P08246 1/20 0.34
USP1 O94782 1/20 0.33
TDP1 Q9NUW8 1/20 0.32
CSNK1D P48730 1/20 0.32
CSNK1E P49674 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9979025 0.81 KCNE1 (0.51) KCNE1CCR1KCNQ1ERCC1FEN1
SCHEMBL6646417 0.77 GAA (0.40) ERCC1FEN1ERCC4RAB9ALIPE
SCHEMBL6645445 0.72 TDP1 (0.50) TP53RAB9AUSP1TDP1
SCHEMBL6645871 0.71 TDP1 (0.44) TP53USP1TDP1
SCHEMBL6649244 0.69 RNASEH1 (0.40) RAB9ATDP1
SCHEMBL6646945 0.69 ERCC1 (0.50) ERCC1FEN1ERCC4
SCHEMBL6883598 0.69 TNKS (0.43) ERCC1FEN1ERCC4
SCHEMBL6885410 0.68 PIN1 (0.60) MAPTERCC1FEN1ERCC4TDP1
SCHEMBL6649378 0.68 ERCC1 (0.58) ERCC1FEN1ERCC4
SCHEMBL6651415 0.68 RIPK1 (0.43) TP53ERCC1FEN1ERCC4RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1819700-A2 POTASSIUM SALT OF AN HIV INTERGRASE INHIBITOR Merck & Co., Inc. (US) 2007-08-22 EP disclosed
WO-2006060712-A9 POTASSIUM SALT OF AN HIV INTEGRASE INHIBITOR MERCK & CO INC (US) 2006-07-27 WO disclosed
WO-2006060712-A2 POTASSIUM SALT OF AN HIV INTEGRASE INHIBITOR MERCK & CO. INC. (US) 2006-06-08 WO disclosed