SCHEMBL5202345

SCHEMBL5202345

Cn1cc(C2CCN(c3c(F)c(F)c(F)c(F)c3C(=O)F)C2)c2ccccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 5/20 0.41
USP2 O75604 1/20 0.40
ALDH1A1 P00352 1/20 0.40
RORC P51449 3/20 0.37
DRD2 P14416 2/20 0.36
SLC6A4 P31645 2/20 0.36
GFER P55789 1/20 0.36
CHRM2 P08172 2/20 0.36
ADRA2A P08913 2/20 0.36
CHRM1 P11229 2/20 0.36
ADRA2B P18089 2/20 0.36
CHRM3 P20309 2/20 0.36
HTR2A P28223 2/20 0.36
HTR2C P28335 2/20 0.36
HTR4 Q13639 2/20 0.36
CYP1A2 P05177 1/20 0.36
CHRM4 P08173 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
ALOX15 P16050 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5202338 0.81 GFER (0.47) HTR6USP2ALDH1A1RORCGFER
SCHEMBL5937364 0.70 ALDH1A1 (0.57) USP2ALDH1A1RORCKDM4ELMNA
SCHEMBL5705162 0.70 RORC (0.51) USP2ALDH1A1RORCCYP1A2CYP2C9
SCHEMBL4859112 0.68 RORC (0.47) HTR6USP2ALDH1A1RORCGFER
SCHEMBL17067795 0.68 ALDH1A1 (0.51) USP2ALDH1A1DRD2SLC6A4HTR2A
SCHEMBL18701720 0.67 RORC (0.49) USP2ALDH1A1RORCKDM4E
SCHEMBL4858049 0.67 MEN1 (0.52) HTR6USP2ALDH1A1RORCCHRM2
SCHEMBL5201722 0.67 HTR2B (0.53) USP2ALDH1A1RORCLMNA
SCHEMBL4858050 0.66 RAB9A (0.62) ALDH1A1RORCKDM4ELMNA
SCHEMBL26912621 0.66 GSK3B (0.46) USP2ALDH1A1DRD2SLC6A4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP claimed