SCHEMBL5202945

SCHEMBL5202945

CC(C)(C)N(Cc1ccc(Oc2ccccc2[N+](=O)[O-])cc1)C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
HTT P42858 1/20 0.48
ESR2 Q92731 1/20 0.45
LMNA P02545 1/20 0.44
LTA4H P09960 1/20 0.44
PTGS1 P23219 1/20 0.44
PTGS2 P35354 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
POLB P06746 2/20 0.43
KDM4E B2RXH2 1/20 0.43
MAPT P10636 1/20 0.43
TDP1 Q9NUW8 2/20 0.43
RXFP1 Q9HBX9 1/20 0.43
SENP8 Q96LD8 1/20 0.43
SENP7 Q9BQF6 1/20 0.43
SENP6 Q9GZR1 1/20 0.43
KMT2A Q03164 3/20 0.42
MEN1 O00255 1/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5206544 0.80 MEN1 (0.45) ALDH1A1HTTLMNAL3MBTL1KMT2A
SCHEMBL5205997 0.78 PTGES (0.45) PTGS1PTGS2POLBMAPTKMT2A
SCHEMBL5201443 0.78 SRD5A2 (0.52) ALDH1A1HTTESR2LTA4HPTGS1
SCHEMBL14674248 0.78 LPAR1 (0.44) LPAR1LPAR5
SCHEMBL5206028 0.77 MAPK1 (0.57) ALDH1A1HTTLMNAL3MBTL1POLB
SCHEMBL5206034 0.77 MAPK1 (0.57) ALDH1A1HTTLMNAL3MBTL1POLB
SCHEMBL5204827 0.76 TDP1 (0.41) HTTLMNAL3MBTL1POLBMAPT
SCHEMBL14674209 0.76 MAPT (0.41) ALDH1A1HTTLMNAPOLBMAPT
SCHEMBL6178891 0.75 HPGD (0.54) ALDH1A1HTTESR2LMNALTA4H
SCHEMBL5204961 0.75 L3MBTL1 (0.51) ALDH1A1HTTLTA4HPTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7160887-B1 Aromatic amine derivatives, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-01-09 US disclosed