SCHEMBL5203471

SCHEMBL5203471

CC(c1ccc(Cl)cc1)C(CNC(=O)C1CCCCN1C)c1ccc(Cl)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.43
CHRNB2 P17787 1/20 0.41
CHRNA5 P30532 1/20 0.41
CHRNA7 P36544 1/20 0.41
CHRNA4 P43681 1/20 0.41
MMP1 P03956 1/20 0.41
MMP3 P08254 1/20 0.41
MMP13 P45452 1/20 0.41
ADAM17 P78536 1/20 0.41
LMNA P02545 1/20 0.41
CCR1 P32246 2/20 0.40
GAA P10253 1/20 0.40
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ALDH1A1 P00352 1/20 0.39
PTGER4 P35408 2/20 0.39
PTGER2 P43116 2/20 0.39
MEN1 O00255 1/20 0.38
MITF O75030 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14064682 0.78 CNR1 (0.48) PTGER4PTGER2
SCHEMBL4829838 0.78 CNR1 (0.48) PTGER4PTGER2
SCHEMBL5201159 0.75 PKM (0.48) LMNAGAAHPGDSMN1; SMN2ALDH1A1
SCHEMBL5261535 0.74 TP53 (0.56) TP53LMNASMN1; SMN2ALDH1A1MEN1
SCHEMBL5266049 0.74 RAB9A (0.60) TP53LMNAHPGDSMN1; SMN2ALDH1A1
Trifluoroacetic Acid SCHEMBL4831463 0.74 CNR1 (0.46)
SCHEMBL21696570 0.73 MEN1 (0.57) ALDH1A1MEN1KMT2A
SCHEMBL5200358 0.73 SMN1; SMN2 (0.41) TP53CCR1GAAHPGDSMN1; SMN2
SCHEMBL4689271 0.72 RAB9A (0.48) LMNAGAAHPGDSMN1; SMN2ALDH1A1
SCHEMBL5200515 0.72 MGLL (0.44) TP53GAAHPGDSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1490043-A4 SPIROCYCLIC AMIDES AS CANNABINOID RECEPTOR MODULATORS MERCK & CO INC (US) 2007-05-30 EP claimed
EP-1490043-A2 SPIROCYCLIC AMIDES AS CANNABINOID RECEPTOR MODULATORS Merck & Co., Inc. (US) 2004-12-29 EP claimed
WO-2003082190-A2 SPIROCYCLIC AMIDES AS CANNABINOID RECEPTOR MODULATORS MERCK & CO., INC. (US) 2003-10-09 WO claimed