SCHEMBL5203532

SCHEMBL5203532

CCOC(=O)[C@H](Cc1ccc2oc(CCCNc3ncc[nH]3)cc(=O)c2c1)NC(=O)OCC(C)(C)C

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 5/20 0.34
ITGAV P06756 5/20 0.34
ITGA2B P08514 1/20 0.33
ALOX15 P16050 1/20 0.33
CTSK P43235 1/20 0.31
TBK1 Q9UHD2 1/20 0.30
ELANE P08246 1/20 0.30
POLB P06746 1/20 0.30
TYR P14679 1/20 0.30
KDM4E B2RXH2 1/20 0.30
LMNA P02545 1/20 0.30
HPGD P15428 1/20 0.30
HSD17B10 Q99714 1/20 0.30
MAOB P27338 1/20 0.30
PRSS1 P07477 1/20 0.30
PRSS2 P07478 1/20 0.30
PRSS3 P35030 1/20 0.30
TPSAB1 Q15661 1/20 0.30
PTGES O14684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14431276 0.93 ITGB3 (0.39) ITGB3ITGAVITGA2BALOX15TYR
SCHEMBL3046466 0.93 ITGB3 (0.39) ITGB3ITGAVITGA2BALOX15TYR
SCHEMBL5207016 0.86 ITGB1 (0.42) ITGB3ITGAVITGA2BTYRKDM4E
SCHEMBL14431257 0.86 ITGB1 (0.42) ITGB3ITGAVITGA2BTYRKDM4E
SCHEMBL5204539 0.86 ITGB3 (0.41) ITGB3ITGAVITGA2BELANEKDM4E
SCHEMBL5206753 0.84 ALOX15 (0.39) ITGB3ITGAVALOX15CTSKTBK1
SCHEMBL5203778 0.83 ITGB3 (0.32) ITGB3ITGAV
SCHEMBL5205119 0.82 ITGB3 (0.38) ITGB3ITGAVALOX15CTSKTBK1
SCHEMBL6495597 0.81 ITGB3 (0.39) ITGB3ITGAVITGA2B
SCHEMBL5208511 0.80 ITGB3 (0.37) ITGB3ITGAVALOX15CTSKTBK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1124824-B1 CHROMENONE AND CHROMANONE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2007-08-22 EP claimed
EP-1124824-B1 CHROMENONE AND CHROMANONE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2007-08-22 EP disclosed
EP-1124824-A1 CHROMENONE AND CHROMANONE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GmbH (DE) 2001-08-22 EP disclosed
WO-2000026212-A1 CHROMENONE AND CHROMANONE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2000-05-11 WO disclosed