SCHEMBL5207016

SCHEMBL5207016

CCOC(=O)[C@H](Cc1ccc2oc(CCCNc3ccccn3)cc(=O)c2c1)NC(=O)OCC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 10/20 0.42
ITGA5 P08648 8/20 0.42
ITGB3 P05106 9/20 0.39
ITGAV P06756 8/20 0.39
MDM4 O15151 1/20 0.38
MDM2 Q00987 1/20 0.38
ITGB5 P18084 2/20 0.35
ITGB6 P18564 2/20 0.35
ITGA2B P08514 3/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
HPGD P15428 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TYR P14679 1/20 0.34
PPARG P37231 1/20 0.33
HDAC4 P56524 1/20 0.33
MEF2D Q14814 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14431257 1.00 ITGB1 (0.42) ITGB1ITGA5ITGB3ITGAVMDM4
SCHEMBL14431255 0.93 ITGB1 (0.50) ITGB1ITGA5ITGB3ITGAVMDM4
SCHEMBL3048694 0.93 ITGB1 (0.50) ITGB1ITGA5ITGB3ITGAVMDM4
SCHEMBL5203532 0.86 ITGB3 (0.34) ITGB3ITGAVITGA2BKDM4ELMNA
SCHEMBL5206753 0.85 ALOX15 (0.39) ITGB3ITGAVKDM4ELMNAHPGD
SCHEMBL5204539 0.84 ITGB3 (0.41) ITGB1ITGA5ITGB3ITGAVITGB5
SCHEMBL5205119 0.83 ITGB3 (0.38) ITGB3ITGAVKDM4ELMNAHPGD
SCHEMBL5210309 0.82 TYR (0.41) ITGB3ITGAVITGA2BKDM4ELMNA
SCHEMBL14431254 0.82 MAPT (0.32) ITGB1ITGA5ITGB3ITGAVKDM4E
SCHEMBL5207840 0.82 MAPT (0.32) ITGB1ITGA5ITGB3ITGAVKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1124824-B1 CHROMENONE AND CHROMANONE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2007-08-22 EP disclosed