SCHEMBL5206753

SCHEMBL5206753

CCOC(=O)[C@H](Cc1ccc2oc(CCCO)cc(=O)c2c1)NC(=O)OCC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.39
ITGB3 P05106 1/20 0.38
ITGAV P06756 1/20 0.38
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36
MAOB P27338 1/20 0.36
TYR P14679 1/20 0.35
STS P08842 2/20 0.35
POLB P06746 3/20 0.34
TBK1 Q9UHD2 1/20 0.34
CTSK P43235 2/20 0.33
PPARG P37231 1/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
THRB P10828 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6498071 0.91 ITGB3 (0.44) ALOX15ITGB3ITGAVTYRSTS
SCHEMBL5205119 0.91 ITGB3 (0.38) ALOX15ITGB3ITGAVKDM4ELMNA
SCHEMBL5208511 0.89 ITGB3 (0.37) ALOX15ITGB3ITGAVKDM4ELMNA
SCHEMBL5210309 0.87 TYR (0.41) ALOX15ITGB3ITGAVKDM4ELMNA
SCHEMBL5207016 0.85 ITGB1 (0.42) ITGB3ITGAVKDM4ELMNAHPGD
SCHEMBL14431257 0.85 ITGB1 (0.42) ITGB3ITGAVKDM4ELMNAHPGD
SCHEMBL5203532 0.84 ITGB3 (0.34) ALOX15ITGB3ITGAVKDM4ELMNA
SCHEMBL3052420 0.83 ITGB3 (0.44) ALOX15ITGB3ITGAVTYRSTS
SCHEMBL6495736 0.82 ITGB3 (0.44) ALOX15ITGB3ITGAVTYRCTSK
SCHEMBL5204539 0.82 ITGB3 (0.41) ITGB3ITGAVKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1124824-B1 CHROMENONE AND CHROMANONE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2007-08-22 EP disclosed
EP-1124824-A1 CHROMENONE AND CHROMANONE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GmbH (DE) 2001-08-22 EP disclosed
WO-2000026212-A1 CHROMENONE AND CHROMANONE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2000-05-11 WO disclosed