Trifluoroacetic Acid

Trifluoroacetic Acid

SCHEMBL5203620

NC(=O)c1nc2c(s1)CCCC2.NCc1cccc(C(=O)N(CC(=O)O)c2ccccc2Cl)c1.O=C(O)C(F)(F)F

nearest known ligand 0.33

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.33
PIK3CB P42338 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
MAPT P10636 3/20 0.32
LMNA P02545 1/20 0.32
GPBAR1 Q8TDU6 1/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
NPSR1 Q6W5P4 1/20 0.31
TPSAB1 Q15661 3/20 0.31
ALDH1A1 P00352 2/20 0.31
POLB P06746 2/20 0.31
NPC1 O15118 2/20 0.30
RAB9A P51151 2/20 0.30
SMN1; SMN2 Q16637 2/20 0.30
PKM P14618 1/20 0.30
FOLH1 Q04609 1/20 0.30
TP53 P04637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5208877 0.95 PIK3CA (0.35) PIK3CAPIK3CBCYP3A4CYP2C9CYP2C19
Trifluoroacetic Acid SCHEMBL5208291 0.85 MAPT (0.33) MAPTLMNATPSAB1NPC1RAB9A
SCHEMBL5210132 0.85 F2 (0.39) MAPTLMNAMEN1KMT2AALDH1A1
Trifluoroacetic Acid SCHEMBL5206023 0.84 ENPP2 (0.36)
Trifluoroacetic Acid SCHEMBL5208518 0.84 FLT3 (0.38) MAPTLMNAMEN1KMT2ANPSR1
Trifluoroacetic Acid SCHEMBL5204591 0.82 F10 (0.33) PIK3CAPIK3CBMAPTGPBAR1KMT2A
SCHEMBL6991435 0.82 F2 (0.35) MAPTLMNAMEN1KMT2AALDH1A1
Trifluoroacetic Acid SCHEMBL5204634 0.81 MAPK10 (0.36) PIK3CAPIK3CBMAPTMEN1KMT2A
Trifluoroacetic Acid SCHEMBL5209006 0.81 PIK3CA (0.33) PIK3CAPIK3CBGPBAR1MEN1KMT2A
Trifluoroacetic Acid SCHEMBL5205966 0.79 PDE4D (0.39) MAPTLMNANPSR1ALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1343561-B1 SERINE PROTEASE INHIBITORS TULARIK LTD (GB) 2007-02-28 EP disclosed
EP-1343561-A1 SERINE PROTEASE INHIBITORS Tularik Limited (GB) 2003-09-17 EP disclosed
WO-2002047762-A1 SERINE PROTEASE INHIBITORS TULARIK LIMITED (GB) 2002-06-20 WO disclosed