SCHEMBL5203686

SCHEMBL5203686

O=C(c1ccc(C(F)(F)F)cc1)N1CCC(c2cn(Cc3ccc4ccccc4c3)c3ccccc23)C1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC5A1 P13866 1/20 0.49
SLC5A2 P31639 1/20 0.49
SLC2A1 P11166 1/20 0.46
HRH3 Q9Y5N1 4/20 0.45
DRD4 P21917 2/20 0.45
HDAC3 O15379 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
NCOR2 Q9Y618 1/20 0.44
ICMT O60725 1/20 0.44
TNF P01375 1/20 0.43
HRH2 P25021 2/20 0.42
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
HTR2B P41595 1/20 0.42
SIGMAR1 Q99720 1/20 0.41
ADRB2 P07550 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5204138 0.89 MGLL (0.49) SLC2A1HRH3HDAC3HDAC1HDAC2
SCHEMBL4862016 0.86 SLC5A1 (0.49) SLC5A1SLC5A2SLC2A1HRH3HDAC3
SCHEMBL4853030 0.86 HDAC3 (0.46) SLC5A1SLC5A2SLC2A1HRH3HDAC3
SCHEMBL5204227 0.85 SLC2A1 (0.46) SLC2A1HDAC3HDAC1HDAC2HDAC10
SCHEMBL5204533 0.85 ALDH1A1 (0.46) HDAC3HDAC1HDAC2HDAC10HDAC8
SCHEMBL3598394 0.84 SIGMAR1 (0.57) SLC2A1HDAC3HDAC1HDAC2HDAC10
SCHEMBL4857565 0.84 HDAC3 (0.46) SLC5A1SLC5A2SLC2A1HDAC3HDAC1
SCHEMBL3605157 0.83 SLC2A1 (0.53) SLC5A1SLC5A2SLC2A1HDAC3HDAC1
SCHEMBL4860077 0.81 SLC2A1 (0.45) SLC5A1SLC5A2SLC2A1HRH3HDAC3
SCHEMBL5204238 0.81 HSD11B1 (0.47) SLC5A1SLC5A2SLC2A1HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP claimed