SCHEMBL5204533

SCHEMBL5204533

CCn1cc(C2CCN(C(=O)c3ccc(C(F)(F)F)cc3)C2)c2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HSD11B1 P28845 2/20 0.46
GAA P10253 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
TPSAB1 Q15661 1/20 0.45
KMT2A Q03164 3/20 0.44
MEN1 O00255 2/20 0.44
HPGD P15428 1/20 0.44
TSHR P16473 1/20 0.44
RAB9A P51151 2/20 0.44
NPC1 O15118 1/20 0.44
ATM Q13315 1/20 0.44
SIGMAR1 Q99720 1/20 0.43
PROKR1 Q8TCW9 1/20 0.42
SLC9A1 P19634 1/20 0.42
MGLL Q99685 1/20 0.42
SMO Q99835 1/20 0.42
MAPK7 Q13164 1/20 0.42
RBP4 P02753 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5203757 0.90 NPC1 (0.57) ALDH1A1SMN1; SMN2HSD11B1TPSAB1KMT2A
SCHEMBL4862016 0.88 SLC5A1 (0.49) ALDH1A1SMN1; SMN2GAASIGMAR1HDAC3
SCHEMBL5204138 0.87 MGLL (0.49) ALDH1A1SMN1; SMN2GAASIGMAR1MGLL
SCHEMBL5202168 0.86 PROKR1 (0.47) ALDH1A1SMN1; SMN2TPSAB1KMT2ARAB9A
SCHEMBL5204500 0.85 TPSAB1 (0.47) ALDH1A1SMN1; SMN2TPSAB1KMT2APROKR1
SCHEMBL5203686 0.85 SLC5A1 (0.49) HSD11B1SIGMAR1HDAC3HDAC1HDAC2
SCHEMBL4862667 0.83 TSHR (0.47) ALDH1A1SMN1; SMN2HSD11B1TPSAB1KMT2A
SCHEMBL3598394 0.83 SIGMAR1 (0.57) HSD11B1GAATDP1KMT2AMEN1
SCHEMBL4853030 0.83 HDAC3 (0.46) ALDH1A1SMN1; SMN2GAASIGMAR1RBP4
SCHEMBL5203268 0.81 GAA (0.48) ALDH1A1SMN1; SMN2HSD11B1GAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP claimed