SCHEMBL5204500

SCHEMBL5204500

CCn1cc(C2CCN(C(=O)c3cc(C(F)(F)F)ccc3Cl)C2)c2ccccc21

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TPSAB1 Q15661 2/20 0.47
KMT2A Q03164 2/20 0.47
ALDH1A1 P00352 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
CRHR1 P34998 3/20 0.46
CRHR2 Q13324 1/20 0.46
HRH2 P25021 1/20 0.42
RORC P51449 3/20 0.42
POLB P06746 1/20 0.42
MAPT P10636 1/20 0.42
MAPK8 P45983 1/20 0.42
MAPK10 P53779 1/20 0.42
PROKR1 Q8TCW9 3/20 0.42
CNR1 P21554 1/20 0.42
HTR6 P50406 1/20 0.41
NR1I2 O75469 1/20 0.41
CACNA1B Q00975 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5203433 0.92 TPSAB1 (0.50) TPSAB1KMT2ACRHR1CRHR2HRH2
SCHEMBL5204533 0.85 ALDH1A1 (0.46) TPSAB1KMT2AALDH1A1SMN1; SMN2HRH2
SCHEMBL4862667 0.82 TSHR (0.47) TPSAB1KMT2AALDH1A1SMN1; SMN2HRH2
SCHEMBL4853030 0.80 HDAC3 (0.46) ALDH1A1SMN1; SMN2HRH2MAPTHTR6
SCHEMBL5202510 0.80 HSD11B1 (0.55) TPSAB1KMT2AALDH1A1SMN1; SMN2HRH2
SCHEMBL5206419 0.80 SMN1; SMN2 (0.49) TPSAB1KMT2AALDH1A1SMN1; SMN2HRH2
SCHEMBL5204238 0.80 HSD11B1 (0.47) KMT2AALDH1A1SMN1; SMN2MAPTHTR6
SCHEMBL5202048 0.78 SLC2A1 (0.44) TPSAB1KMT2AALDH1A1SMN1; SMN2MAPT
SCHEMBL5202100 0.78 ALDH1A1 (0.51) TPSAB1KMT2AALDH1A1SMN1; SMN2HRH2
SCHEMBL5202168 0.78 PROKR1 (0.47) TPSAB1KMT2AALDH1A1SMN1; SMN2HRH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP claimed
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP disclosed