SCHEMBL5205017

SCHEMBL5205017

O=C(O)Cc1ccc(NS(=O)(=O)c2ccccc2)cc1

nearest known ligand 0.75

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 5/20 0.75
HDAC8 Q9BY41 3/20 0.75
ALDH1A1 P00352 4/20 0.67
POLB P06746 1/20 0.67
GAA P10253 1/20 0.64
MEN1 O00255 3/20 0.62
KMT2A Q03164 3/20 0.62
HDAC4 P56524 1/20 0.62
KDM4E B2RXH2 1/20 0.62
PKM P14618 1/20 0.62
HTR6 P50406 1/20 0.62
KEAP1 Q14145 2/20 0.61
IL1RN P18510 1/20 0.61
ERAP1 Q9NZ08 1/20 0.61
CASP6 P55212 1/20 0.59
PTGDR2 Q9Y5Y4 1/20 0.58
LMNA P02545 1/20 0.58
FABP4 P15090 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27889027 0.93 ALDH1A1 (0.67) HDAC1HDAC8ALDH1A1POLBGAA
SCHEMBL5202198 0.87 HDAC1 (0.71) HDAC1HDAC8ALDH1A1GAAMEN1
SCHEMBL27884380 0.86 KMT2A (0.61) HDAC1HDAC8ALDH1A1POLBGAA
SCHEMBL8074277 0.86 ALDH1A1 (0.74) HDAC1HDAC8ALDH1A1POLBGAA
SCHEMBL14812106 0.86 HDAC8 (1.00) HDAC1HDAC8ALDH1A1MEN1KMT2A
SCHEMBL397676 0.84 HDAC1 (0.68) HDAC1HDAC8ALDH1A1POLBMEN1
SCHEMBL27430787 0.84 PGR (0.71) HDAC1HDAC8ALDH1A1POLBGAA
SCHEMBL8249490 0.84 HDAC1 (0.76) HDAC1HDAC8ALDH1A1POLBMEN1
SCHEMBL31681345 0.83 ALDH1A1 (0.63) HDAC1HDAC8ALDH1A1POLBGAA
SCHEMBL2822371 0.83 MEN1 (0.67) HDAC1HDAC8ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 41 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070197437-A1 COMPOSITIONS FOR ENHANCED EPITHELIAL PERMEATION OF Y2 RECEPTOR-BINDING PEPTIDES NASTECH PHARMACEUTICAL COMPANY INC. 2007-08-23 US disclosed
US-20070161563-A1 A DEVICE FOR ENHANCED EPITHELIAL PERMEATION OF Y2 RECEPTOR-BINDING PEPTIDES NASTECH PHARMACEUTICAL COMPANY INC. 2007-07-12 US disclosed
US-7229966-B2 Compositions and methods for enhanced mucosal delivery of Y2 receptor-binding peptides and methods for treating and preventing obesity NASTECH PHARMACEUTICAL COMPANY INC. (US) 2007-06-12 US disclosed
US-20070129299-A1 COMPOSITIONS AND METHODS FOR ENHANCED MUCOSAL DELIVERY OF PYY PEPTIDE NASTECH PHARMACEUTICAL COMPANY INC. 2007-06-07 US disclosed
US-7186691-B2 Compositions and methods for enhanced mucosal delivery of Y2 receptor-binding peptides and methods for treating and preventing obesity NASTECH PHARMACEUTICAL COMPANY INC. (US) 2007-03-06 US disclosed
US-7160887-B1 Aromatic amine derivatives, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-01-09 US disclosed
US-7157426-B2 such as peptide YY, Neuropeptide Y, or Pancreatic polypeptide with solubilizing agent (cyclodextran), chelating agent (ethylenediamine tetraacetic acid), and polyol such as sucrose NASTECH PHARMACEUTICAL COMPANY INC. (US) 2007-01-02 US disclosed
US-20060134130-A1 Oral drug delivery compositions and methods EMISPHERE TECHNOLOGIES, INC. (US) 2006-06-22 US disclosed
US-7005141-B2 Oral drug delivery compositions and methods EMISPHERE TECHNOLOGIES INC. (US) 2006-02-28 US disclosed
CN-1726044-A Compositions and methods for enhancing mucosal delivery of Y2 receptor-binding peptides and methods for treating and preventing obesity NASTECH PHARM CO (US) 2006-01-25 CN disclosed
US-5766633-A MODIFIED AMINO ACID CARRIER, BIOACTIVE PEPTIDES EMISPHERE TECHNOLOGIES, INC. (US) 1998-06-16 US disclosed
US-5709861-A PEPTIDES WITH ANTIGENS AND PROCESS FOR MIXING EMISPHERE TECHNOLOGIES, INC. (US) 1998-01-20 US disclosed
EP-0812212-A1 COMPOSITIONS FOR THE DELIVERY OF ANTIGENS Emisphere Technologies, Inc. (US) 1997-12-17 EP disclosed
EP-0784469-A1 COMPOSITIONS FOR THE DELIVERY OF ANTIGENS Emisphere Technologies, Inc. (US) 1997-07-23 EP disclosed
EP-0696208-A4 ORAL DRUG DELIVERY COMPOSITIONS AND METHODS EMISPHERE TECH INC (US) 1997-01-29 EP disclosed
WO-1996021464-A9 COMPOSITIONS FOR THE DELIVERY OF ANTIGENS 1996-11-14 WO disclosed
WO-1996021464-A1 COMPOSITIONS FOR THE DELIVERY OF ANTIGENS EMISPHERE TECHNOLOGIES, INC. (US) 1996-07-18 WO disclosed
WO-1996012474-A1 COMPOSITIONS FOR THE DELIVERY OF ANTIGENS EMISPHERE TECHNOLOGIES, INC. (US) 1996-05-02 WO disclosed
EP-0696208-A1 ORAL DRUG DELIVERY COMPOSITIONS AND METHODS Emisphere Technologies, Inc. (US) 1996-02-14 EP disclosed
WO-1994023767-A1 ORAL DRUG DELIVERY COMPOSITIONS AND METHODS EMISPHERE TECHNOLOGIES, INC. (US) 1994-10-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060134130-A1 Oral drug delivery compositions and methods ADM2, PTMS, DNPEP HDAC1 2962/4885HDAC8 1441/4885ALDH1A1 3433/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.