SCHEMBL5205026

SCHEMBL5205026

O=C(O)Cc1ccccc1NS(=O)(=O)c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.58
KDM4E B2RXH2 1/20 0.58
PTGDR2 Q9Y5Y4 1/20 0.53
CXCL8 P10145 3/20 0.51
KMT2A Q03164 4/20 0.51
TSHR P16473 2/20 0.51
RECQL P46063 2/20 0.50
POLB P06746 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
SQSTM1 Q13501 1/20 0.49
KEAP1 Q14145 1/20 0.49
NFE2L2 Q16236 1/20 0.49
DPP4 P27487 1/20 0.49
PTGS2 P35354 2/20 0.49
AKR1B10 O60218 1/20 0.49
UGT1A9 O60656 1/20 0.49
TRPA1 O75762 1/20 0.49
ABCB11 O95342 1/20 0.49
MT-CO2 P00403 1/20 0.49
TTR P02766 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7866143 0.90 LMNA (0.59) ALDH1A1KDM4EPTGDR2KMT2ATSHR
SCHEMBL16397682 0.86 BCL2 (0.55) ALDH1A1KDM4EPTGDR2KMT2ATSHR
SCHEMBL398529 0.84 KMT2A (0.47) ALDH1A1KDM4EPTGDR2KMT2ATSHR
SCHEMBL3897238 0.84 KEAP1 (0.55) ALDH1A1KDM4EKMT2ATSHRPOLB
SCHEMBL12050285 0.83 RECQL (0.57) ALDH1A1KDM4EKMT2ATSHRRECQL
SCHEMBL3563417 0.82 PTGDR2 (0.56) ALDH1A1KDM4EPTGDR2KMT2ATSHR
SCHEMBL7888388 0.81 PTGS2 (0.54) ALDH1A1KDM4ECXCL8KMT2AKEAP1
SCHEMBL10272404 0.81 ALDH1A1 (0.71) ALDH1A1KMT2ATSHRRECQLPOLB
SCHEMBL21647703 0.81 PTGDR2 (0.49) ALDH1A1KDM4EPTGDR2KMT2ATSHR
SCHEMBL7425678 0.80 ALDH1A1 (0.55) ALDH1A1KDM4EKMT2ATSHRSQSTM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7160887-B1 Aromatic amine derivatives, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-01-09 US disclosed
EP-1123918-B1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME TAKEDA PHARMACEUTICAL (JP) 2005-03-09 EP disclosed
EP-1123918-A1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME Takeda Chemical Industries, Ltd. (JP) 2001-08-16 EP disclosed