SCHEMBL5205166

SCHEMBL5205166

CCOC(=O)CN(Cc1ccccc1)C(=O)[C@@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(C)C

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 4/20 0.48
CTSL P07711 1/20 0.41
CTSB P07858 1/20 0.41
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41
ELANE P08246 1/20 0.41
KMT2A Q03164 2/20 0.40
PIN1 Q13526 1/20 0.40
MDM4 O15151 1/20 0.39
TP53 P04637 1/20 0.39
TNF P01375 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27571135 1.00 CASP3 (0.48) CASP3CTSLCTSBCTSSCTSK
SCHEMBL27561296 0.94 CASP3 (0.44) CASP3CTSLCTSBCTSSCTSK
SCHEMBL5201715 0.94 CASP3 (0.44) CASP3CTSLCTSBCTSSCTSK
SCHEMBL5201718 0.94 CASP3 (0.44) CASP3CTSLCTSBCTSSCTSK
SCHEMBL5201071 0.90 CASP3 (0.53) CASP3CTSLCTSBCTSSCTSK
SCHEMBL5200510 0.88 PTPN1 (0.44) CASP3CTSLCTSBCTSSCTSK
SCHEMBL27561654 0.88 PTPN1 (0.44) CASP3CTSLCTSBCTSSCTSK
SCHEMBL7325639 0.84 CTSL (0.57) CTSLCTSBCTSSCTSKELANE
SCHEMBL22457336 0.80 CASP3 (0.45) CASP3KMT2APIN1MDM4TP53
SCHEMBL21313691 0.80 CASP3 (0.56) CASP3KMT2APIN1MDM4TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1400521-B1 PIPERAZINE COMPOUNDS KOWA CO (JP) 2007-11-07 EP disclosed
EP-1400521-A1 PIPERAZINE COMPOUNDS Kowa Co., Ltd. (JP) 2004-03-24 EP disclosed
US-6432957-B1 ANTIASTHMA; ANTIALLERGENS; RHEUMATIC DISEASES; ANTIINFLAMMATORY AGENTS KOWA CO., LTD. (JP) 2002-08-13 US disclosed