SCHEMBL5206090

SCHEMBL5206090

Nc1ncc(Oc2ccc(F)cc2Cl)c(NCCO)n1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BCL6 P41182 3/20 0.42
SLC6A2 P23975 2/20 0.39
SLC6A3 Q01959 2/20 0.39
SLC6A4 P31645 1/20 0.37
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
STK17B O94768 2/20 0.35
STK17A Q9UEE5 2/20 0.35
SLC22A12 Q96S37 1/20 0.35
CCNT1 O60563 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
SCN9A Q15858 1/20 0.35
P2RX3 P56373 1/20 0.34
P2RX2 Q9UBL9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5203455 0.88 TTR (0.40) BCL6SLC6A2SLC6A3SLC6A4CYP2D6
SCHEMBL5207181 0.84 BCL6 (0.40) BCL6SLC6A2SLC6A3SLC6A4CYP2D6
SCHEMBL5207953 0.80 SLC6A2 (0.44) SLC6A2SLC6A3SLC6A4CYP2C19ALDH1A1
SCHEMBL7513223 0.77 CCNT1 (0.37) BCL6CYP2D6CYP2C19STK17BSTK17A
SCHEMBL5205013 0.77 KCNH2 (0.40) CYP2D6CYP2C19STK17ACCNT1ALDH1A1
SCHEMBL7161091 0.76 MAPK14 (0.43) CCNT1
SCHEMBL7161086 0.76 MAPK14 (0.43) CCNT1
SCHEMBL5203877 0.76 NPC1 (0.36) SLC6A2SLC6A3SLC6A4SLC22A12SCN9A
SCHEMBL7716686 0.72 HTR3E (0.42) SLC6A4MAPTSCN9A
SCHEMBL5205294 0.72 MMP13 (0.40) ALDH1A1MAPTSCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165523-B1 NEUROTROPHIC SUBSTITUTED PYRIMIDINES KRENITSKY PHARMACEUTICALS INC (US) 2007-11-07 EP claimed
EP-1165523-B1 NEUROTROPHIC SUBSTITUTED PYRIMIDINES KRENITSKY PHARMACEUTICALS INC (US) 2007-11-07 EP disclosed
US-6916820-B1 Neurotrophic substituted pyrimidines KRENITSKY PHARMACEUTICALS, INC. (US) 2005-07-12 US disclosed