SCHEMBL5206471

SCHEMBL5206471

Cc1cc(Cc2cnc[nH]2)cc(NS(C)(=O)=O)c1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.54
ADRA1A P35348 1/20 0.54
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
HRH3 Q9Y5N1 8/20 0.41
HRH4 Q9H3N8 3/20 0.41
TAAR1 Q96RJ0 1/20 0.41
LMNA P02545 1/20 0.40
MAPT P10636 2/20 0.40
CYP3A4 P08684 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PTGS1 P23219 1/20 0.39
PDPK1 O15530 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5204050 0.75 ADRA1A (0.42) ADRA2AADRA1AHRH3HRH4MAPT
SCHEMBL5203578 0.75 ADRA1A (0.53) ADRA2AADRA1AHRH3HRH4TAAR1
SCHEMBL16882475 0.72 HPGD (0.44) CYP11B1CYP11B2LMNAMAPTCYP3A4
Oxalic Acid SCHEMBL5200567 0.71 ADRA1A (0.38) ADRA2AADRA1AHRH3HRH4MAPT
SCHEMBL12865227 0.70 TOP2A (0.50) CYP11B1CYP11B2LMNAMAPTCYP3A4
SCHEMBL5204185 0.70 HTR1D (0.49) ADRA2AADRA1AHRH3TAAR1LMNA
SCHEMBL12865204 0.69 KEAP1 (0.50) LMNAMAPTSMN1; SMN2PTGS1ALDH1A1
SCHEMBL3267511 0.69 PTGS1 (0.50) LMNAMAPTSMN1; SMN2PTGS1ALDH1A1
SCHEMBL5201429 0.68 ADRA1A (0.48) ADRA2AADRA1AHRH3HRH4TAAR1
SCHEMBL7595633 0.67 LMNA (0.74) LMNAMAPTSMN1; SMN2ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0887346-B1 N-Phenyl-alkylsulfonamide derivatives, their preparation and their use as alpha1A/1L adrenoceptor agonists HOFFMANN LA ROCHE (CH) 2007-12-12 EP disclosed