SCHEMBL5223490

SCHEMBL5223490

CCCN1CCN(Cc2cnn(-c3ccc(-c4ccc(F)cc4)cc3)c2-c2ccoc2)CC1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMO Q99835 3/20 0.40
MAPT P10636 3/20 0.38
DRD2 P14416 4/20 0.38
DRD4 P21917 4/20 0.38
DRD3 P35462 4/20 0.38
LMNA P02545 3/20 0.36
L3MBTL1 Q9Y468 3/20 0.36
NPC1 O15118 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ALDH1A1 P00352 2/20 0.34
POLB P06746 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5227160 0.92 SMO (0.41) SMOMAPTDRD2DRD4DRD3
SCHEMBL5224829 0.89 SMO (0.42) SMOMAPTDRD2DRD4DRD3
SCHEMBL5224226 0.82 L3MBTL1 (0.36) SMOMAPTDRD2DRD4DRD3
SCHEMBL5224144 0.80 HTR2C (0.38) SMOMAPT
SCHEMBL5225265 0.79 SMO (0.59) SMOMAPTDRD2DRD4DRD3
SCHEMBL5228311 0.78 NR3C1 (0.34) SMOLMNANPC1HPGDTSHR
SCHEMBL5222796 0.78 NR3C1 (0.35) SMOLMNANPC1RAB9ASMN1; SMN2
SCHEMBL5228124 0.76 SMO (0.43) SMOMAPTDRD2DRD4DRD3
SCHEMBL2761009 0.75 SMO (0.43) SMOMAPTDRD2DRD4DRD3
SCHEMBL2761237 0.75 SMO (0.43) SMOMAPTDRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed