SCHEMBL5222796

SCHEMBL5222796

CN(C)Cc1cnn(-c2ccc(-c3ccc(F)cc3)cc2)c1-c1ccoc1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 6/20 0.35
LMNA P02545 2/20 0.35
ALDH1A1 P00352 2/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
SMO Q99835 2/20 0.35
PTGS2 P35354 1/20 0.34
NPSR1 Q6W5P4 1/20 0.33
PGR P06401 2/20 0.33
KCNH2 Q12809 1/20 0.33
MAPK1 P28482 1/20 0.32
ACHE P22303 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CLK4 Q9HAZ1 1/20 0.31
NR3C2 P08235 1/20 0.31
P2RX7 Q99572 1/20 0.31
S1PR1 P21453 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5228311 0.89 NR3C1 (0.34) NR3C1LMNAALDH1A1NPC1RAB9A
SCHEMBL5224670 0.80 NR3C1 (0.35) NR3C1LMNAALDH1A1NPC1RAB9A
SCHEMBL5227160 0.79 SMO (0.41) LMNAALDH1A1SMOCYP1A2CYP3A4
SCHEMBL5223490 0.78 SMO (0.40) LMNAALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL5225124 0.76 PIK3CD (0.42) NR3C1LMNAALDH1A1NPC1RAB9A
SCHEMBL5224829 0.75 SMO (0.42) LMNAALDH1A1SMN1; SMN2SMOMAPK1
SCHEMBL5224144 0.74 HTR2C (0.38) NR3C1SMO
SCHEMBL5224226 0.73 L3MBTL1 (0.36) NR3C1ALDH1A1SMOKCNH2
SCHEMBL5227271 0.72 DHODH (0.39) NR3C1LMNAALDH1A1SMN1; SMN2PGR
SCHEMBL5227418 0.72 PTGS1 (0.38) NR3C1LMNAALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed