SCHEMBL5228311

SCHEMBL5228311

CCN(CC)Cc1cnn(-c2ccc(-c3ccc(F)cc3)cc2)c1-c1ccoc1

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 6/20 0.34
TP53 P04637 2/20 0.34
SMO Q99835 2/20 0.34
NPC1 O15118 3/20 0.33
LMNA P02545 3/20 0.33
RAB9A P51151 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
ALDH1A1 P00352 1/20 0.32
PGR P06401 2/20 0.32
CYP17A1 P05093 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5222796 0.89 NR3C1 (0.35) NR3C1SMONPC1LMNARAB9A
SCHEMBL5232217 0.78 NR3C1 (0.40) NR3C1TP53NPC1RAB9APGR
SCHEMBL5223490 0.78 SMO (0.40) SMONPC1LMNARAB9ASMN1; SMN2
SCHEMBL5227160 0.78 SMO (0.41) SMOLMNACYP1A2CYP2C19ALDH1A1
SCHEMBL5228140 0.77 NR3C1 (0.48) NR3C1TP53SMOLMNARAB9A
SCHEMBL5224829 0.74 SMO (0.42) SMOLMNASMN1; SMN2ALDH1A1
SCHEMBL5228824 0.73 ICMT (0.40) NR3C1TP53LMNASMN1; SMN2HPGD
SCHEMBL5224144 0.72 HTR2C (0.38) NR3C1SMO
SCHEMBL5230496 0.72 PTGS1 (0.37) NR3C1TP53SMONPC1LMNA
SCHEMBL5224226 0.72 L3MBTL1 (0.36) NR3C1TP53SMOTSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed