SCHEMBL5223850

SCHEMBL5223850

COc1cccc(CCNC[C@@H](O)[C@H](Cc2ccccc2)N(C(=O)O)C(C)(C)C)c1OC

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSG P08311 1/20 0.48
CMA1 P23946 1/20 0.48
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 1/20 0.42
TAAR1 Q96RJ0 1/20 0.42
BCHE P06276 6/20 0.42
BACE1 P56817 1/20 0.41
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA14 Q9ULX7 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
ITGA4 P13612 1/20 0.39
ITGB7 P26010 1/20 0.39
ADRB2 P07550 1/20 0.39
ADRB1 P08588 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5223861 1.00 CTSG (0.48) CTSGCMA1KDM4EALDH1A1TAAR1
SCHEMBL5226954 0.92 OPRM1 (0.47) KDM4EALDH1A1TAAR1BCHEBACE1
SCHEMBL5226961 0.92 OPRM1 (0.47) KDM4EALDH1A1TAAR1BCHEBACE1
SCHEMBL5223889 0.83 ALDH1A1 (0.38) ALDH1A1BCHEBACE1OPRM1OPRD1
SCHEMBL5223892 0.83 ALDH1A1 (0.38) ALDH1A1BCHEBACE1OPRM1OPRD1
SCHEMBL5219646 0.83 ADRB3 (0.43) KDM4EBCHEBACE1OPRM1OPRD1
SCHEMBL5219638 0.83 ADRB3 (0.43) KDM4EBCHEBACE1OPRM1OPRD1
SCHEMBL5217626 0.83 SIGMAR1 (0.43) OPRM1KMT2A
SCHEMBL5217634 0.83 SIGMAR1 (0.43) OPRM1KMT2A
SCHEMBL5216394 0.82 OPRM1 (0.47) KDM4EALDH1A1BCHEBACE1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567488-B1 HYDROXYETHYLAMINE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE GLAXO GROUP LTD (GB) 2007-02-21 EP disclosed