SCHEMBL5225128

SCHEMBL5225128

Cc1noc(C)c1-c1[nH]ncc1C(c1ccc(-c2ccc(F)cc2)cc1)N(C)C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NSD3 Q9BZ95 1/20 0.45
GPR55 Q9Y2T6 1/20 0.44
BRD4 O60885 11/20 0.41
CREBBP Q92793 2/20 0.39
PTGS2 P35354 2/20 0.35
USP2 O75604 2/20 0.34
LMNA P02545 2/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2C19 P33261 2/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
ALOX15 P16050 1/20 0.34
APEX1 P27695 1/20 0.34
KMT2A Q03164 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TP53 P04637 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
HIF1A Q16665 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5223627 0.79 GPR55 (0.42) NSD3GPR55BRD4CREBBPLMNA
SCHEMBL5228026 0.79 HTR1A (0.42) NSD3GPR55BRD4CREBBPCYP1A2
SCHEMBL5224159 0.79 GPR55 (0.43) NSD3GPR55BRD4CREBBPUSP2
SCHEMBL5225734 0.76 GPR55 (0.39) NSD3GPR55BRD4CREBBP
SCHEMBL16404607 0.68 BRD4 (0.66) GPR55BRD4PTGS2USP2LMNA
SCHEMBL2001308 0.67 CYP17A1 (0.36) MEN1ALDH1A1KMT2ACYP3A4
SCHEMBL5553073 0.65 BRD4 (0.53) GPR55BRD4CREBBPLMNACYP1A2
SCHEMBL20148798 0.61 MAPK14 (0.50) LMNAKMT2A
SCHEMBL1998048 0.60 MAPT (0.36) USP2LMNAMEN1ALDH1A1KMT2A
SCHEMBL5228222 0.60 HRH3 (0.39) CYP2C19CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed