SCHEMBL5225734

SCHEMBL5225734

Cc1noc(C)c1-c1[nH]ncc1C(c1ccc(-c2ccc(F)cc2)cc1)N1CCC(O)C1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GPR55 Q9Y2T6 1/20 0.39
NSD3 Q9BZ95 1/20 0.39
BRD4 O60885 17/20 0.38
CREBBP Q92793 1/20 0.36
RORC P51449 1/20 0.35
BRD2 P25440 1/20 0.34
BRD3 Q15059 1/20 0.34
BRDT Q58F21 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5224159 0.85 GPR55 (0.43) GPR55NSD3BRD4CREBBPBRD2
SCHEMBL5228026 0.85 HTR1A (0.42) GPR55NSD3BRD4CREBBPBRD2
SCHEMBL2001557 0.83 KCNH2 (0.37)
SCHEMBL5223627 0.83 GPR55 (0.42) GPR55NSD3BRD4CREBBP
SCHEMBL5227625 0.79 HTR7 (0.37)
SCHEMBL5228031 0.78 MAPK1 (0.40)
SCHEMBL5225128 0.76 NSD3 (0.45) GPR55NSD3BRD4CREBBP
SCHEMBL5907357 0.76 HTR1A (0.39)
SCHEMBL2000118 0.75 KCNH2 (0.33)
SCHEMBL2003026 0.74 GSK3B (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed