SCHEMBL5228026

SCHEMBL5228026

Cc1noc(C)c1-c1[nH]ncc1C(c1ccc(-c2ccc(F)cc2)cc1)N1CCNCC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.42
HTR7 P34969 3/20 0.42
HTR2B P41595 3/20 0.42
HTR6 P50406 3/20 0.42
NSD3 Q9BZ95 1/20 0.41
GPR55 Q9Y2T6 1/20 0.41
P4HB P07237 1/20 0.41
HTR1D P28221 2/20 0.40
HTR3A P46098 1/20 0.40
BRD4 O60885 11/20 0.38
BRD2 P25440 2/20 0.38
BRD3 Q15059 2/20 0.38
CREBBP Q92793 1/20 0.37
CYP1A2 P05177 3/20 0.36
HSD17B10 Q99714 1/20 0.36
HTR1B P28222 1/20 0.35
HTR5A P47898 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP3A4 P08684 1/20 0.34
HIF1A Q16665 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5224159 0.90 GPR55 (0.43) NSD3GPR55BRD4BRD2CREBBP
SCHEMBL5223627 0.89 GPR55 (0.42) NSD3GPR55BRD4CREBBPCYP1A2
SCHEMBL5225734 0.85 GPR55 (0.39) NSD3GPR55BRD4BRD2BRD3
SCHEMBL5225128 0.79 NSD3 (0.45) NSD3GPR55BRD4CREBBPCYP1A2
SCHEMBL5228222 0.73 HRH3 (0.39) HTR1AHTR7HTR2BHTR6P4HB
SCHEMBL1997982 0.70 ACHE (0.43) HTR1AHTR2BP4HB
SCHEMBL2761010 0.69 MAPT (0.41) HTR1AHTR7HTR2BHTR6P4HB
SCHEMBL2761138 0.69 LMNA (0.40) HTR1AHTR7HTR2BHTR6P4HB
SCHEMBL2004264 0.69 HTR1A (0.41) HTR1AHTR7HTR2BHTR6P4HB
SCHEMBL1998316 0.68 HRH3 (0.45) HTR1AHTR2BP4HBCYP1A2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed