SCHEMBL5224159

SCHEMBL5224159

Cc1noc(C)c1-c1[nH]ncc1C(c1ccc(-c2ccc(F)cc2)cc1)N1CCN(C)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR55 Q9Y2T6 1/20 0.43
NSD3 Q9BZ95 1/20 0.41
BRD4 O60885 10/20 0.38
ACHE P22303 3/20 0.37
CREBBP Q92793 2/20 0.37
BRD2 P25440 1/20 0.36
ALDH1A1 P00352 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36
LMNA P02545 1/20 0.36
TSHR P16473 1/20 0.36
HIF1A Q16665 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
DRD2 P14416 1/20 0.35
DRD4 P21917 1/20 0.35
DRD3 P35462 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
USP2 O75604 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5223627 0.90 GPR55 (0.42) GPR55NSD3BRD4ACHECREBBP
SCHEMBL5228026 0.90 HTR1A (0.42) GPR55NSD3BRD4CREBBPBRD2
SCHEMBL5225734 0.85 GPR55 (0.39) GPR55NSD3BRD4CREBBPBRD2
SCHEMBL5228222 0.84 HRH3 (0.39) ACHETSHRDRD2DRD4DRD3
SCHEMBL1997982 0.81 ACHE (0.43) ACHETSHRDRD3HRH3CYP2D6
SCHEMBL2761010 0.79 MAPT (0.41) ACHECYP3A4LMNADRD2DRD4
SCHEMBL5225128 0.79 NSD3 (0.45) GPR55NSD3BRD4CREBBPALDH1A1
SCHEMBL5230180 0.77 HTR1A (0.42) ACHEALDH1A1CYP3A4LMNATSHR
SCHEMBL2761124 0.74 BCL2L11 (0.40) LMNATSHR
SCHEMBL5907425 0.73 CHRM2 (0.43) ALDH1A1CYP3A4LMNATSHRDRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed