SCHEMBL5225924

SCHEMBL5225924

COC(=O)CN(Cc1ccc(O)cc1)S(=O)(=O)N1CCCC1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TAS2R14 Q9NYV8 4/20 0.40
TSHR P16473 3/20 0.40
PTPN1 P18031 2/20 0.39
LMNA P02545 1/20 0.38
ALDH1A1 P00352 4/20 0.38
HSD17B10 Q99714 1/20 0.38
SCN3A Q9NY46 1/20 0.38
TDP1 Q9NUW8 1/20 0.37
PKM P14618 1/20 0.36
CYP3A4 P08684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5435181 0.90 TAS2R14 (0.39) TAS2R14TSHRPTPN1ALDH1A1TDP1
SCHEMBL5313019 0.89 ALDH1A1 (0.44) TAS2R14LMNAALDH1A1
SCHEMBL5225058 0.84 ALDH1A1 (0.54) PTPN1LMNAALDH1A1
SCHEMBL5434168 0.76 ALDH1A1 (0.53) PTPN1LMNAALDH1A1HSD17B10
SCHEMBL5224874 0.75 ALDH1A1 (0.52) PTPN1ALDH1A1
SCHEMBL5225370 0.74 PPARG (0.52)
SCHEMBL2513385 0.72 TAS2R14 (0.70) TAS2R14PTPN1ALDH1A1
SCHEMBL10958880 0.66 NR1D1 (0.51) PTPN1LMNAALDH1A1HSD17B10
SCHEMBL6177245 0.65 MTOR (0.50) TSHRPTPN1ALDH1A1
SCHEMBL4540959 0.65 MEN1 (0.64) TAS2R14PTPN1ALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070254882-A1 Sulfamide Derivatives and Pharmaceutical Composition for Upregulation of Lipid Metabolism Comprising Same CRYSTAL GENOMICS, INC. (KR) 2007-11-01 US disclosed
EP-1778654-A1 SULFAMIDE DERIVATIVES AND PHARMACEUTICAL COMPOSITION FOR UPREGULATION OF LIPID METABOLISM COMPRISING SAME Crystalgenomics, Inc. (KR) 2007-05-02 EP disclosed
WO-2006006832-A1 SULFAMIDE DERIVATIVES AND PHARMACEUTICAL COMPOSITION FOR UPREGULATION OF LIPID METABOLISM COMPRISING SAME CRYSTALGENOMICS, INC. (KR) 2006-01-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070254882-A1 Sulfamide Derivatives and Pharmaceutical Composition for Upregulation of Lipid Metabolism Comprising Same SULT2A1, SPTLC2, SGMS2 TAS2R14 502/4885TSHR 2726/4885PTPN1 1365/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.