SCHEMBL5226450

SCHEMBL5226450

OC1CCN(Cc2cnn(-c3ccc(C4=C(Cc5ccccc5)OCO4)cc3)c2-c2ccco2)C1

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
F10 P00742 15/20 0.35
F2 P00734 12/20 0.35
ALDH1A1 P00352 1/20 0.33
NPC1 O15118 1/20 0.33
KMT2A Q03164 1/20 0.33
LTA4H P09960 1/20 0.33
PDCD1 Q15116 1/20 0.33
CD274 Q9NZQ7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5229345 0.89 EGFR (0.34) ALDH1A1KMT2A
SCHEMBL5222928 0.85 SMO (0.38) ALDH1A1KMT2A
SCHEMBL5226173 0.85 SMO (0.38) ALDH1A1NPC1KMT2A
SCHEMBL5226844 0.85 SIGMAR1 (0.34) ALDH1A1KMT2A
SCHEMBL5226667 0.85 DRD4 (0.39) ALDH1A1KMT2A
SCHEMBL5225471 0.82 HRH3 (0.35) LTA4HCD274
SCHEMBL5230408 0.81 SLC2A1 (0.32) ALDH1A1PDCD1CD274
SCHEMBL5226446 0.81 ALDH1A1 (0.41) ALDH1A1NPC1KMT2APDCD1CD274
SCHEMBL5229304 0.80 ALDH1A1 (0.33) ALDH1A1
SCHEMBL5228505 0.79 F10 (0.48) F10F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed