SCHEMBL5229345

SCHEMBL5229345

NC1CCN(Cc2cnn(-c3ccc(C4=C(Cc5ccccc5)OCO4)cc3)c2-c2ccco2)CC1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.34
ERBB2 P04626 2/20 0.34
SMO Q99835 3/20 0.33
DRD2 P14416 1/20 0.33
DRD4 P21917 1/20 0.33
DRD3 P35462 1/20 0.33
ALDH1A1 P00352 4/20 0.33
AAK1 Q2M2I8 3/20 0.33
USP2 O75604 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
TSHR P16473 1/20 0.33
HCRTR1 O43613 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
KDM4E B2RXH2 2/20 0.32
MAPT P10636 2/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5226450 0.89 F10 (0.35) ALDH1A1KMT2A
SCHEMBL5226173 0.88 SMO (0.38) SMODRD2DRD4DRD3ALDH1A1
SCHEMBL5226844 0.88 SIGMAR1 (0.34) SMODRD2DRD4DRD3ALDH1A1
SCHEMBL5222928 0.88 SMO (0.38) SMODRD2DRD4DRD3ALDH1A1
SCHEMBL5226667 0.88 DRD4 (0.39) SMODRD2DRD4DRD3ALDH1A1
SCHEMBL5225471 0.84 HRH3 (0.35) SMODRD2DRD4DRD3KDM4E
SCHEMBL5230408 0.83 SLC2A1 (0.32) EGFRERBB2ALDH1A1TSHRHCRTR1
SCHEMBL5229304 0.81 ALDH1A1 (0.33) ALDH1A1USP2TSHRSMN1; SMN2LMNA
SCHEMBL5229335 0.80 ALDH1A1 (0.42) ALDH1A1AAK1USP2MEN1KMT2A
SCHEMBL5224860 0.80 ALDH1A1 (0.31) ALDH1A1TSHRLMNAKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed