SCHEMBL5226512

SCHEMBL5226512

O=C(Nc1nnn[nH]1)Oc1cccs1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 1/20 0.40
MMP2 P08253 1/20 0.40
MMP9 P14780 1/20 0.40
MMP12 P39900 1/20 0.40
ALDH1A1 P00352 4/20 0.34
NPC1 O15118 5/20 0.33
LMNA P02545 3/20 0.33
HTT P42858 3/20 0.33
NPSR1 Q6W5P4 2/20 0.33
GMNN O75496 1/20 0.33
ABL1 P00519 1/20 0.33
TUBB4A P04350 1/20 0.33
TP53 P04637 1/20 0.33
CYP1A2 P05177 1/20 0.33
TUBB P07437 1/20 0.33
TUBA3C P0DPH7 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C9 P11712 1/20 0.33
TSHR P16473 1/20 0.33
NFKB1 P19838 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL896715 0.78 F2 (0.47) ALDH1A1LMNAHTTTP53CYP1A2
SCHEMBL9138103 0.77 ALDH1A1 (0.56) ALDH1A1NPC1LMNAHTTTP53
SCHEMBL13715730 0.75 NPC1 (0.54) ALDH1A1NPC1LMNAHTTTP53
SCHEMBL9756827 0.72 ALDH1A1 (0.41) ALDH1A1NPC1LMNAHTTMAPT
SCHEMBL9756826 0.71 RAB9A (0.60) ALDH1A1NPC1LMNAHTTTP53
SCHEMBL1480730 0.71 KDM4E (0.39) ALDH1A1NPC1LMNAHTTABL1
SCHEMBL20894431 0.71 NPC1 (0.58) ALDH1A1NPC1LMNANPSR1TP53
SCHEMBL28007813 0.70 SMN1; SMN2 (0.51) ALDH1A1NPC1HTTTP53MAPT
SCHEMBL9088000 0.70
SCHEMBL15559316 0.69 MGLL (0.46) ALDH1A1NPC1NPSR1MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1636212-B1 CYCLOALKYLSULFANYL SUBSTITUTED BENZO¬B|THIOPHENES AS THERAPEUTIC AGENTS WARNER LAMBERT CO (US) 2007-06-27 EP claimed