SCHEMBL5226913

SCHEMBL5226913

Fc1ccc(-c2ccc(C(c3cn[nH]c3-c3cccc(Cl)c3)N3CCN(C4CCCC4)CC3)cc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 8/20 0.45
TSHR P16473 5/20 0.42
ALDH1A1 P00352 4/20 0.41
NPSR1 Q6W5P4 1/20 0.41
CCR5 P51681 1/20 0.40
KDM2B Q8NHM5 1/20 0.39
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
HTR1A P08908 2/20 0.39
HTR2A P28223 2/20 0.39
HTR7 P34969 2/20 0.39
HTR2B P41595 2/20 0.39
HTR3A P46098 2/20 0.39
HTR6 P50406 2/20 0.39
HTR2C P28335 1/20 0.39
HTR5A P47898 1/20 0.39
MEN1 O00255 1/20 0.39
PKM P14618 1/20 0.39
KMT2A Q03164 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5230180 0.86 HTR1A (0.42) HRH3TSHRALDH1A1HTR1AHTR2A
SCHEMBL5230614 0.85 ACHE (0.51) HRH3HTR1AHTR2AHTR7HTR2B
SCHEMBL5227779 0.85 ACHE (0.52) HRH3CNR1CNR2HTR1AHTR2A
SCHEMBL5227450 0.84 HRH3 (0.42) HRH3ALDH1A1NPSR1HTR1AHTR2A
SCHEMBL5228031 0.83 MAPK1 (0.40) CNR1CNR2HTR1AHTR2AHTR7
SCHEMBL2761178 0.81 TSHR (0.48) HRH3TSHRALDH1A1NPSR1CCR5
SCHEMBL5229632 0.79 HTR2A (0.40) HTR1AHTR2AHTR7HTR2BHTR3A
SCHEMBL5907344 0.72 MAPK1 (0.41) HRH3CNR1CNR2HTR1AHTR2A
SCHEMBL2761079 0.71 TSHR (0.40) HRH3TSHRALDH1A1NPSR1CCR5
SCHEMBL5226495 0.70 NPSR1 (0.44) HRH3TSHRALDH1A1NPSR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed