SCHEMBL5230865

SCHEMBL5230865

COc1cccc2[nH]cc(C(C)(CC(N)=O)C3CCCCC3)c12

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.41
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40
SCN5A Q14524 1/20 0.37
SCN2A Q99250 1/20 0.37
HTR6 P50406 1/20 0.37
ADRB2 P07550 1/20 0.37
DRD2 P14416 2/20 0.36
DRD4 P21917 2/20 0.36
DRD3 P35462 2/20 0.36
ICMT O60725 1/20 0.36
ALDH1A1 P00352 2/20 0.35
HPGD P15428 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35
POLB P06746 1/20 0.35
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5319290 0.74 HTR2A (0.41) HTR2AHTR2CHTR2BMTNR1AMTNR1B
SCHEMBL3160107 0.70 MTNR1A (0.33) HTR2AHTR2CHTR2BMTNR1AMTNR1B
SCHEMBL5230871 0.67 HTR2A (0.45) HTR2AHTR2CHTR2BMTNR1AMTNR1B
SCHEMBL5102654 0.66 HTR2A (0.52) HTR2AHTR2CHTR2BMTNR1AMTNR1B
SCHEMBL31181454 0.65 HTR2A (0.46) HTR2AHTR2CHTR2BMTNR1AMTNR1B
SCHEMBL5202202 0.65 HTR6 (0.56) HTR2AHTR2CHTR2BMTNR1AMTNR1B
SCHEMBL3943593 0.64 MAPT (0.39) HTR2AHTR2CHTR2BMTNR1AMTNR1B
SCHEMBL5202211 0.64 MTNR1A (0.52) HTR2AMTNR1AMTNR1BSCN5ASCN2A
SCHEMBL2071662 0.64 MTNR1A (0.42) HTR2AHTR2CHTR2BMTNR1AMTNR1B
SCHEMBL788913 0.62 HTR2A (0.57) HTR2AHTR2CHTR2BMTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1756054-A1 3-AMINO-1-ARYLPROPYL INDOLES AS MONOAMINE REUPTAKE INHIBITOR F.HOFFMANN-LA ROCHE AG (CH) 2007-02-28 EP disclosed
WO-2005118539-A1 3-AMINO-1-ARYLPROPYL INDOLES AS MONOAMINE REUPTAKE INHIBITOR F.HOFFMANN-LA ROCHE AG (CH) 2005-12-15 WO disclosed