SCHEMBL5233120

SCHEMBL5233120

Cc1cccc(C(=O)Cc2ccnc3ccc(OC(F)(F)F)cc23)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.44
TGFBR1 P36897 1/20 0.44
PTGS2 P35354 2/20 0.40
PTGS1 P23219 1/20 0.40
WNT3A P56704 1/20 0.40
TP53 P04637 1/20 0.39
MTNR1A P48039 3/20 0.39
MTNR1B P49286 3/20 0.39
SCN10A Q9Y5Y9 1/20 0.38
KDM4C Q9H3R0 1/20 0.38
BRAF P15056 1/20 0.37
RAF1 P04049 1/20 0.37
LCK P06239 1/20 0.37
RET P07949 1/20 0.37
CYP3A4 P08684 1/20 0.37
KIT P10721 1/20 0.37
KDR P35968 1/20 0.37
MAP3K20 Q9NYL2 1/20 0.37
RIPK3 Q9Y572 1/20 0.37
MMP13 P45452 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23851296 0.87 MTNR1A (0.52) TGFBR1MTNR1AMTNR1B
SCHEMBL31461239 0.87 MTNR1A (0.52) TGFBR1MTNR1AMTNR1B
SCHEMBL4873486 0.86 SMN1; SMN2 (0.47) TGFBR1TP53MTNR1AMTNR1B
SCHEMBL5239692 0.84 TGFBR1 (0.41) TGFBR1BRAFKDRMAP3K20DHODH
SCHEMBL24322279 0.83 CDK8 (0.39) TGFBR1DHODH
SCHEMBL3747756 0.81 ALDH1A1 (0.39) TGFBR1TP53CYP3A4KDRPTGFR
SCHEMBL31461243 0.81 ALDH1A1 (0.39) TGFBR1TP53CYP3A4KDRPTGFR
SCHEMBL5235225 0.80 CYP1A2 (0.49) TGFBR1CYP3A4
SCHEMBL29959459 0.80 CYP1A2 (0.49) TGFBR1CYP3A4
SCHEMBL5235795 0.80 KDR (0.45) TGFBR1MTNR1AMTNR1BRETKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397364-B1 NOVEL PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS LILLY CO ELI (US) 2007-07-25 EP disclosed