SCHEMBL5236574

SCHEMBL5236574

O=C(Cc1ccnc2cc(Cl)ccc12)c1ccccn1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.48
PRNP P04156 2/20 0.46
RXFP1 Q9HBX9 2/20 0.46
KDM4E B2RXH2 1/20 0.46
KMT2A Q03164 3/20 0.45
POLB P06746 1/20 0.45
AGTR1 P30556 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
GRM5 P41594 1/20 0.45
CHKA P35790 1/20 0.44
GRM4 Q14833 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
NR4A2 P43354 2/20 0.43
SOS2 Q07890 1/20 0.43
PKM P14618 1/20 0.43
CYP1A2 P05177 1/20 0.43
BACE1 P56817 1/20 0.42
LMNA P02545 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5231726 0.84 GRM4 (0.44) KDM4EKMT2AL3MBTL1GRM5GRM4
SCHEMBL4872056 0.83 CYP1A2 (0.55) KDM4EKMT2AL3MBTL1GRM4CYP1A2
SCHEMBL5231489 0.83 PRNP (0.45) PRNPRXFP1KDM4EKMT2APOLB
SCHEMBL5233929 0.81 CYP1A2 (0.50) TSHRKMT2AL3MBTL1CYP1A2SMN1; SMN2
SCHEMBL5232920 0.81 RAB9A (0.49) KDM4EKMT2AL3MBTL1GRM5GRM4
SCHEMBL5231287 0.80 NPC1 (0.49) KDM4EKMT2APOLBL3MBTL1GRM4
SCHEMBL5233499 0.78 GRM4 (0.43) KDM4EKMT2AL3MBTL1GRM5GRM4
SCHEMBL5238508 0.77 CYP1A2 (0.49) KMT2ACYP1A2SMN1; SMN2
SCHEMBL5235583 0.75 KDM5A (0.48) TSHRKDM4EKMT2AL3MBTL1GRM5
SCHEMBL5239810 0.74 THRB (0.40) TSHRKDM4EKMT2ACHKAPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397364-B1 NOVEL PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS LILLY CO ELI (US) 2007-07-25 EP disclosed