SCHEMBL5236705

SCHEMBL5236705

CNC1(CC=O)CN(c2ccc(-c3ccc(OC)c(F)c3)cc2)CCN1C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 1/20 0.41
FFAR4 Q5NUL3 1/20 0.37
FFAR1 O14842 1/20 0.37
ERN1 O75460 1/20 0.36
PDE4B Q07343 1/20 0.36
ALDH1A1 P00352 4/20 0.36
HPGD P15428 1/20 0.36
MAPK1 P28482 1/20 0.36
LCK P06239 1/20 0.35
MAP4K3 Q8IVH8 1/20 0.35
MAP4K1 Q92918 1/20 0.35
CYP17A1 P05093 1/20 0.35
TP53 P04637 1/20 0.35
TDP2 O95551 1/20 0.35
MAPT P10636 4/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
HTR1A P08908 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5236271 0.88 ERN1 (0.43) FFAR1ERN1ALDH1A1MAPK1TP53
SCHEMBL5234847 0.85 KMT2A (0.40) ALDH1A1HPGDTP53MAPTHTR1A
SCHEMBL5239486 0.84 FGFR1 (0.41) ERN1ALDH1A1HPGDMAPK1MAPT
SCHEMBL5236555 0.83 USP2 (0.41) FFAR4ALDH1A1HPGDMAPK1TP53
SCHEMBL5233074 0.82 L3MBTL1 (0.44) ALDH1A1MAPK1MAPTHTR1ALMNA
SCHEMBL5232294 0.82 ALDH1A1 (0.39) ALDH1A1HPGDTP53MAPTHTR1A
SCHEMBL5236699 0.81 CD274 (0.41) CD274FFAR4FFAR1PDE4BALDH1A1
SCHEMBL5233790 0.81 CA2 (0.38) CD274MAPTLMNA
SCHEMBL5237663 0.80 KCNA5 (0.37) FFAR4CYP3A4
SCHEMBL5232205 0.80 SLC6A7 (0.41) ALDH1A1HPGDMAPTLMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1701946-B1 DERIVATIVES OF 1-PIPERAZINE- AND 1-HOMOPIPERAZINE-CARBOXYLATES, PREPARATION METHOD THEREOF AND USE OF SAME AS INHIBITORS OF THE FAAH ENZYME SANOFI AVENTIS (FR) 2007-12-19 EP claimed