SCHEMBL5237698

SCHEMBL5237698

CC(C)n1c(=O)n(C)c(=O)c2c1ncn2CCO

nearest known ligand 0.72

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 8/20 0.72
LMNA P02545 3/20 0.72
PDE4A P27815 3/20 0.64
PDE4B Q07343 3/20 0.64
PDE4C Q08493 3/20 0.64
PDE4D Q08499 3/20 0.64
SMN1; SMN2 Q16637 2/20 0.56
POLB P06746 1/20 0.53
MAPT P10636 1/20 0.52
ADORA2A P29274 2/20 0.51
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
MAPK1 P28482 1/20 0.49
RXFP1 Q9HBX9 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5272670 0.92 PDE4A (0.65) ADORA2BLMNAPDE4APDE4BPDE4C
SCHEMBL5275531 0.91 PDE4A (0.60) ADORA2BLMNAPDE4APDE4BPDE4C
Etofylline SCHEMBL149271 0.84 ADORA2B (1.00) ADORA2BLMNAPDE4APDE4BPDE4C
SCHEMBL28752095 0.81 ALDH1A1 (0.75) ADORA2BLMNASMN1; SMN2POLBRXFP1
SCHEMBL556077 0.79 SMN1; SMN2 (0.74) ADORA2BLMNASMN1; SMN2POLBMAPK1
SCHEMBL11366248 0.77 PDE4A (0.58) ADORA2BLMNAPDE4APDE4BPDE4C
SCHEMBL9293406 0.75 ADORA2B (0.83) ADORA2BLMNAPDE4APDE4BPDE4C
SCHEMBL20011104 0.74 LMNA (0.62) ADORA2BLMNASMN1; SMN2POLBMAPT
SCHEMBL8697228 0.74 ADORA2B (0.81) ADORA2BLMNAPDE4APDE4BPDE4C
SCHEMBL11359942 0.74 RXFP1 (0.67) ADORA2BLMNAPDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1829523-A1 Cosmetic use of an N-oxide derivative of theophylline L'OREAL (FR) 2007-09-05 EP disclosed