SCHEMBL5239241

SCHEMBL5239241

CC(=O)Nc1ccc(C(=O)N2CC3CN(c4cccc(CCC(N)=O)c4)CC3C2)cc1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.43
CYP2C19 P33261 1/20 0.40
CYP2C9 P11712 1/20 0.39
TSHR P16473 1/20 0.39
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
KDM4C Q9H3R0 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
GRIN2B Q13224 1/20 0.38
NAMPT P43490 3/20 0.37
POLB P06746 2/20 0.37
MAPT P10636 1/20 0.37
TP53 P04637 1/20 0.36
HPGD P15428 1/20 0.36
AOC3 Q16853 1/20 0.36
LMNA P02545 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
SIRT1 Q96EB6 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5230954 0.91 GABRD (0.42) HTTTSHRALDH1A1KDM4ENAMPT
SCHEMBL5237823 0.90 SLC6A7 (0.36) HTTNAMPTMAPTHPGDLMNA
SCHEMBL5232788 0.86 CHRNB2 (0.44) TSHRPOLBMAPTLMNA
SCHEMBL5231026 0.84 HPGD (0.42) HTTALDH1A1NAMPTHPGDLMNA
SCHEMBL5237286 0.83 LMNA (0.43) HTTALDH1A1LMNA
SCHEMBL5233538 0.83 ALDH1A1 (0.47) HTTTSHRALDH1A1POLBTP53
SCHEMBL4694593 0.83 ALDH1A1 (0.41) ALDH1A1KDM4ETDP1HPGD
SCHEMBL5236638 0.82 ALDH1A1 (0.44) CYP2C19CYP2C9ALDH1A1
SCHEMBL5237460 0.82 PLA2G10 (0.39) ALDH1A1HPGDAOC3
SCHEMBL5238361 0.82 HPGD (0.43) HTTTDP1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed