SCHEMBL5248346

SCHEMBL5248346

CCNC(=O)c1ccc(-n2cc(C(=O)NCc3cccc(OCC)c3)nn2)c(OCCOCCF)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 3/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2D6 P10635 2/20 0.45
CYP2C9 P11712 2/20 0.45
ROCK1 Q13464 2/20 0.45
POLB P06746 1/20 0.43
LMNA P02545 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
BRD4 O60885 2/20 0.40
GLS O94925 3/20 0.40
DDT P30046 3/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
CHRM3 P20309 1/20 0.39
PSEN1 P49768 1/20 0.39
PSEN2 P49810 1/20 0.39
APH1B Q8WW43 1/20 0.39
NCSTN Q92542 1/20 0.39
APH1A Q96BI3 1/20 0.39
PSENEN Q9NZ42 1/20 0.39
KLKB1 P03952 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5244747 0.94 BRD4 (0.47) ROCK2CYP3A4CYP2D6CYP2C9ROCK1
SCHEMBL5248746 0.93 ROCK2 (0.43) ROCK2CYP3A4CYP2D6CYP2C9ROCK1
SCHEMBL5244551 0.93 ROCK2 (0.45) ROCK2CYP3A4CYP2D6CYP2C9ROCK1
SCHEMBL5246370 0.92 GLS (0.51) ROCK2ROCK1GLS
SCHEMBL5246709 0.91 ROCK2 (0.42) ROCK2ROCK1POLBLMNABRD4
SCHEMBL5246767 0.91 MIF (0.47) CYP2D6CYP2C9LMNAL3MBTL1BRD4
SCHEMBL5246245 0.90 ROCK2 (0.41) ROCK2ROCK1BRD4DDTPSEN1
SCHEMBL5246030 0.90 LMNA (0.42) ROCK2ROCK1POLBLMNABRD4
SCHEMBL5249644 0.89 LOX (0.40) ROCK2CYP3A4CYP2D6CYP2C9ROCK1
SCHEMBL5248515 0.89 DDT (0.39) ROCK2ROCK1BRD4GLSDDT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1867331-A1 TRIAZOLE DERIVATIVE AND THE USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-12-19 EP disclosed