SCHEMBL5249644

SCHEMBL5249644

CCNC(=O)c1ccc(-n2cc(C(=O)NCc3cccc(Oc4ccccn4)c3)nn2)c(OCCOCCF)c1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LOX P28300 3/20 0.40
LOXL2 Q9Y4K0 3/20 0.40
GLS O94925 3/20 0.38
BRD4 O60885 2/20 0.37
ROCK2 O75116 2/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2D6 P10635 2/20 0.37
CYP2C9 P11712 2/20 0.37
ROCK1 Q13464 2/20 0.37
DDT P30046 3/20 0.37
PSEN1 P49768 2/20 0.37
PSEN2 P49810 2/20 0.37
APH1B Q8WW43 2/20 0.37
NCSTN Q92542 2/20 0.37
APH1A Q96BI3 2/20 0.37
PSENEN Q9NZ42 2/20 0.37
MIF P14174 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5246605 0.92 LOX (0.39) LOXLOXL2GLSDDTPSEN1
SCHEMBL5244747 0.89 BRD4 (0.47) GLSBRD4ROCK2CYP3A4CYP2D6
SCHEMBL5248346 0.89 ROCK2 (0.45) GLSBRD4ROCK2CYP3A4CYP2D6
SCHEMBL5244551 0.88 ROCK2 (0.45) GLSBRD4ROCK2CYP3A4CYP2D6
SCHEMBL5246767 0.88 MIF (0.47) GLSBRD4CYP2D6CYP2C9DDT
SCHEMBL5246370 0.87 GLS (0.51) GLSROCK2ROCK1
SCHEMBL5246709 0.86 ROCK2 (0.42) GLSBRD4ROCK2ROCK1DDT
SCHEMBL5244330 0.86 BRD4 (0.42) LOXLOXL2BRD4DDTPSEN1
SCHEMBL5246245 0.86 ROCK2 (0.41) BRD4ROCK2ROCK1DDTPSEN1
SCHEMBL5246030 0.86 LMNA (0.42) BRD4ROCK2ROCK1DDTPSEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1867331-A1 TRIAZOLE DERIVATIVE AND THE USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-12-19 EP disclosed