SCHEMBL5251920

SCHEMBL5251920

COC(=O)C(=O)c1c(C2CC2)[nH]c2ccccc12

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TUBB4A P04350 2/20 0.54
TUBB P07437 2/20 0.54
TUBA3C P0DPH7 2/20 0.54
TUBA1B P68363 2/20 0.54
TUBA4A P68366 2/20 0.54
TUBB4B P68371 2/20 0.54
TUBB3 Q13509 2/20 0.54
TUBB2A Q13885 2/20 0.54
TUBB8 Q3ZCM7 2/20 0.54
TUBA3E Q6PEY2 2/20 0.54
TUBA1A Q71U36 2/20 0.54
TUBA1C Q9BQE3 2/20 0.54
TUBB6 Q9BUF5 2/20 0.54
TUBB2B Q9BVA1 2/20 0.54
TUBB1 Q9H4B7 2/20 0.54
NR4A2 P43354 2/20 0.48
NPC1 O15118 2/20 0.47
RAB9A P51151 1/20 0.47
KDM4E B2RXH2 3/20 0.44
HSD17B10 Q99714 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4984795 0.82 TUBB4A (0.49) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL6438378 0.80 L3MBTL1 (0.47) NPC1RAB9AKDM4EKMT2AALDH1A1
SCHEMBL4561758 0.78 NR4A2 (0.71) NR4A2NPC1RAB9AHSD17B10HTT
SCHEMBL14367890 0.77 ALDH1A1 (0.59) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL8352535 0.77 NR4A2 (0.72) NR4A2RAB9AKDM4EHSD17B10MEN1
SCHEMBL14440308 0.77 NR4A2 (0.53) NR4A2KDM4EHSD17B10MEN1KMT2A
SCHEMBL5257370 0.74 NR4A2 (0.50) NR4A2KDM4EHSD17B10MEN1KMT2A
SCHEMBL6990972 0.72 NR4A2 (0.48) NR4A2RAB9AKDM4EHSD17B10TSHR
SCHEMBL5143038 0.71 KDM4E (0.51) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL28296520 0.70 BRD3 (0.47) TUBB4ATUBBTUBA3CTUBA1BTUBA4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487822-B1 PYRROLE-2,5-DIONE DERIVATIVES AND THEIR USE AS GSK-3 INHIBITORS LILLY CO ELI (US) 2007-08-01 EP disclosed
CN-1639152-A Pyrrole-2, 5-dione derivatives and their use as GSK-3 inhibitors LILLY CO ELI (US) 2005-07-13 CN disclosed