SCHEMBL5263996

SCHEMBL5263996

CC(c1ccc(Cl)cc1)C(CNC(=O)c1cc2ccccc2o1)c1ccc(Cl)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP24A1 Q07973 3/20 0.59
TDP1 Q9NUW8 2/20 0.57
TP53 P04637 3/20 0.52
ALDH1A1 P00352 3/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
HPGD P15428 1/20 0.51
LMNA P02545 1/20 0.51
THRB P10828 1/20 0.51
NPC1 O15118 4/20 0.50
RAB9A P51151 4/20 0.50
L3MBTL1 Q9Y468 2/20 0.50
KDM4E B2RXH2 1/20 0.50
TSHR P16473 1/20 0.50
NFKB1 P19838 1/20 0.50
NFKB2 Q00653 1/20 0.50
RELA Q04206 1/20 0.50
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
ATM Q13315 1/20 0.49
TAS1R3 Q7RTX0 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5373381 0.79 UTS2R (0.55) TDP1SMN1; SMN2NPC1RAB9AMEN1
SCHEMBL5262685 0.79 KDM4E (0.47) CYP24A1TDP1TP53SMN1; SMN2LMNA
SCHEMBL5263994 0.79 NPC1 (0.60) CYP24A1TDP1TP53ALDH1A1SMN1; SMN2
SCHEMBL5261415 0.78 P2RX7 (0.46) SMN1; SMN2NPC1RAB9ATSHRMEN1
SCHEMBL5095558 0.78 SMN1; SMN2 (0.63) TP53ALDH1A1SMN1; SMN2HPGDLMNA
SCHEMBL5262774 0.78 SLC6A9 (0.54) TP53SMN1; SMN2NPC1RAB9AKDM4E
Hydrochloric Acid SCHEMBL5551493 0.77 ALDH1A1 (0.62) TP53ALDH1A1SMN1; SMN2HPGDLMNA
Hydrochloric Acid SCHEMBL5551489 0.77 ALDH1A1 (0.62) TP53ALDH1A1SMN1; SMN2HPGDLMNA
SCHEMBL5266049 0.76 RAB9A (0.60) TP53ALDH1A1SMN1; SMN2HPGDLMNA
SCHEMBL5552009 0.76 ALDH1A1 (0.60) TP53ALDH1A1SMN1; SMN2HPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1494997-A4 SUBSTITUTED ARYL AMIDES MERCK & CO INC (US) 2007-04-11 EP disclosed
EP-1494997-A1 SUBSTITUTED ARYL AMIDES Merck & Co., Inc. (US) 2005-01-12 EP disclosed
WO-2003087037-A1 SUBSTITUTED ARYL AMIDES MERCK & CO., INC. (US) 2003-10-23 WO disclosed