SCHEMBL5267623

SCHEMBL5267623

CCc1cccc(C(=O)Cc2ccnc3cc(Cl)c(Cl)cc23)n1

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 4/20 0.37
PTGER1 P34995 9/20 0.35
CBLB Q13191 1/20 0.35
CYP1A2 P05177 3/20 0.34
CYP2C9 P11712 2/20 0.34
NR1H4 Q96RI1 1/20 0.33
KDM4E B2RXH2 1/20 0.32
MAPT P10636 1/20 0.32
CLK1 P49759 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29959944 0.84 CYP1A2 (0.47) CYP1A2
SCHEMBL5234356 0.84 CYP1A2 (0.47) CYP1A2
SCHEMBL5237932 0.75 CYP1A2 (0.48) CYP1A2KDM4E
SCHEMBL5231489 0.74 PRNP (0.45) MRGPRX4CYP1A2KDM4ECLK1
SCHEMBL5234890 0.72 P2RX7 (0.39) CYP1A2KDM4E
SCHEMBL4872415 0.72 CYP1A2 (0.49) CYP1A2KDM4EMAPTCLK1
SCHEMBL5231308 0.70 SRC (0.42)
SCHEMBL5231071 0.70 MEN1 (0.36) PTGER1CYP1A2CYP2C9MAPT
SCHEMBL6671176 0.70 NPC1 (0.40)
SCHEMBL4490632 0.70 P2RX7 (0.39) CYP1A2KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1543001-B1 PYRAZOLOPYRIDINE DERIVATIVES AS TGF BETA SIGNAL TRANSDUCTION INHIBITORS FOR THE TREATMENT OF CANCER LILLY CO ELI (US) 2007-08-15 EP disclosed