SCHEMBL5268784

SCHEMBL5268784

O=C(NC1CCCC1)c1n[nH]cc1NS(=O)(=O)c1cccc2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
EPHX2 P34913 1/20 0.45
LMNA P02545 1/20 0.44
EPHX1 P07099 2/20 0.43
PLA2G7 Q13093 6/20 0.42
HIF1A Q16665 1/20 0.42
KCNA5 P22460 2/20 0.41
TSHR P16473 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
ALDH1A1 P00352 2/20 0.40
HTT P42858 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
KDM4E B2RXH2 1/20 0.40
NR1I2 O75469 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5274014 0.85 ALDH1A1 (0.54) LMNAKCNA5TSHRMEN1KMT2A
SCHEMBL5270919 0.83 KCNA5 (0.51) KCNA5TSHRMEN1KMT2AALDH1A1
SCHEMBL5269930 0.83 KCNA5 (0.47) KCNA5TSHRMEN1KMT2AALDH1A1
SCHEMBL5270560 0.83 LMNA (0.54) NPC1RAB9ALMNAKCNA5ALDH1A1
SCHEMBL5270515 0.82 EPHX1 (0.46) NPC1RAB9AEPHX2LMNAEPHX1
SCHEMBL5268522 0.82 LMNA (0.48) NPC1RAB9ALMNAEPHX1KCNA5
SCHEMBL5273547 0.81 TSHR (0.49) LMNAKCNA5TSHRMEN1KMT2A
SCHEMBL5265874 0.79 SLC16A3 (0.48) KCNA5TSHRMEN1KMT2AALDH1A1
SCHEMBL5269318 0.79 LMNA (0.53) NPC1RAB9ALMNAKCNA5MEN1
SCHEMBL5268725 0.79 RAB9A (0.51) NPC1RAB9AKCNA5TSHRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1847531-A1 PYRAZOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2007-10-24 EP disclosed