SCHEMBL5265874

SCHEMBL5265874

O=C(NCc1ccccc1)c1n[nH]cc1NS(=O)(=O)c1cccc2ccccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC16A3 O15427 3/20 0.48
KCNA5 P22460 1/20 0.47
TSHR P16473 1/20 0.45
CCKBR P32239 1/20 0.44
F2 P00734 2/20 0.42
PRSS1 P07477 2/20 0.42
PRSS2 P07478 2/20 0.42
PRSS3 P35030 2/20 0.42
MCL1 Q07820 1/20 0.42
NPY5R Q15761 1/20 0.42
PGR P06401 1/20 0.42
KDM4E B2RXH2 1/20 0.42
GSK3B P49841 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
HCRTR1 O43613 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HTT P42858 1/20 0.41
PFKFB3 Q16875 1/20 0.41
ACLY P53396 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5268725 0.91 RAB9A (0.51) SLC16A3KCNA5TSHRCCKBRMCL1
SCHEMBL5270341 0.87 MEN1 (0.54) SLC16A3KCNA5MEN1KMT2AALDH1A1
SCHEMBL5268835 0.86 HPGD (0.52) TSHRKDM4EMEN1KMT2AALDH1A1
SCHEMBL5273547 0.85 TSHR (0.49) SLC16A3KCNA5TSHRPGRMEN1
SCHEMBL5269930 0.84 KCNA5 (0.47) SLC16A3KCNA5TSHRPGRMEN1
SCHEMBL5268485 0.84 KCNA5 (0.51) KCNA5KDM4EMEN1KMT2AALDH1A1
SCHEMBL5270919 0.83 KCNA5 (0.51) SLC16A3KCNA5TSHRMCL1PGR
SCHEMBL5268920 0.82 KCNA5 (0.47) SLC16A3KCNA5MCL1MEN1KMT2A
SCHEMBL5266632 0.82 CASP1 (0.42) KDM4EGSK3BKMT2AALDH1A1
SCHEMBL5268993 0.81 ALDH1A1 (0.54) TSHRKDM4EKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1847531-A1 PYRAZOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2007-10-24 EP disclosed