SCHEMBL5269930

SCHEMBL5269930

CNC(=O)c1n[nH]cc1NS(=O)(=O)c1cccc2ccccc12

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 1/20 0.47
HCRTR1 O43613 1/20 0.47
TSHR P16473 1/20 0.45
USP2 O75604 1/20 0.45
USP8 P40818 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
EDNRA P25101 3/20 0.43
EDNRB P24530 2/20 0.43
SLC16A3 O15427 4/20 0.43
PGR P06401 1/20 0.43
PGAM1 P18669 1/20 0.42
PLK1 P53350 1/20 0.42
ALDH1A1 P00352 1/20 0.41
HTT P42858 1/20 0.41
PFKFB3 Q16875 1/20 0.41
ACLY P53396 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5270919 0.89 KCNA5 (0.51) KCNA5HCRTR1TSHRUSP2USP8
SCHEMBL5273547 0.86 TSHR (0.49) KCNA5HCRTR1TSHRUSP2USP8
SCHEMBL5265874 0.84 SLC16A3 (0.48) KCNA5HCRTR1TSHRMEN1KMT2A
SCHEMBL5267782 0.83 GAA (0.55) KCNA5TSHRMEN1KMT2AALDH1A1
SCHEMBL5268784 0.83 NPC1 (0.47) KCNA5TSHRMEN1KMT2AALDH1A1
SCHEMBL5268725 0.82 RAB9A (0.51) KCNA5TSHRMEN1KMT2ASLC16A3
SCHEMBL5318573 0.80 SLC40A1 (0.49) KCNA5TSHRMEN1KMT2AALDH1A1
SCHEMBL5268835 0.80 HPGD (0.52) TSHRMEN1KMT2AALDH1A1HTT
SCHEMBL5271876 0.79 MTNR1A (0.43) PGRPLK1ALDH1A1
SCHEMBL5269789 0.79 MEN1 (0.51) TSHRMEN1KMT2APGRPGAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1847531-A1 PYRAZOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2007-10-24 EP disclosed