SCHEMBL5269732

SCHEMBL5269732

CC(C)NC(=O)c1n[nH]cc1NS(=O)(=O)C(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.40
CYP1A2 P05177 1/20 0.40
ADORA3 P0DMS8 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA2B P29275 1/20 0.34
ADORA1 P30542 1/20 0.34
KDM4E B2RXH2 1/20 0.34
DYRK1A Q13627 5/20 0.34
MEN1 O00255 1/20 0.34
POLB P06746 1/20 0.34
KMT2A Q03164 1/20 0.34
BRD4 O60885 1/20 0.33
MLKL Q8NB16 1/20 0.33
MLYCD O95822 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
ALOX15 P16050 1/20 0.32
TSHR P16473 1/20 0.32
CASP1 P29466 1/20 0.32
ADRA1D P25100 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5269326 0.87 KDM4E (0.42) SMN1; SMN2CYP1A2ADORA3ADORA2AADORA2B
SCHEMBL5265886 0.83 LMNA (0.45) SMN1; SMN2CYP1A2KDM4EMEN1KMT2A
SCHEMBL5267963 0.81 MLKL (0.43) SMN1; SMN2CYP1A2MEN1KMT2AMLKL
SCHEMBL5266813 0.80 MEN1 (0.35) SMN1; SMN2MEN1POLBKMT2ABRD4
SCHEMBL5265268 0.80 KCNA5 (0.46) SMN1; SMN2CYP1A2ADORA3ADORA2AADORA2B
SCHEMBL13816853 0.80 SMN1; SMN2 (0.44) SMN1; SMN2CYP1A2ADORA3ADORA2AADORA2B
SCHEMBL5270110 0.79 KCNK3 (0.42) SMN1; SMN2CYP1A2KDM4EBRD4
SCHEMBL5271810 0.79 KCNA5 (0.50) SMN1; SMN2KDM4EPOLBTSHR
SCHEMBL5265233 0.79 ALDH1A1 (0.44) SMN1; SMN2ADORA2AKDM4EPOLBKMT2A
SCHEMBL5269256 0.78 TSHR (0.44) SMN1; SMN2CYP1A2MEN1POLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1847531-A1 PYRAZOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2007-10-24 EP disclosed