SCHEMBL5280260

SCHEMBL5280260

O=C(O)Cc1cc(Br)c(Oc2cc(Br)c(O)c(Br)c2)c(Br)c1

nearest known ligand 0.68

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
THRB P10828 20/20 0.68
THRA P10827 17/20 0.68
PPARG P37231 2/20 0.68
ITGB3 P05106 1/20 0.55
ITGAV P06756 1/20 0.55
RXRA P19793 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5858355 0.84 THRB (0.56) THRBTHRAPPARG
SCHEMBL5283381 0.83 THRA (0.52) THRBTHRAPPARGITGB3ITGAV
SCHEMBL5278593 0.83 THRB (0.80) THRBTHRAPPARG
SCHEMBL5859452 0.81 THRB (0.62) THRBTHRAPPARG
SCHEMBL5287547 0.79 THRB (0.73) THRBTHRAPPARG
SCHEMBL5279787 0.78 THRB (0.74) THRBTHRAPPARG
SCHEMBL7220499 0.78 THRB (0.69) THRBTHRAPPARG
SCHEMBL5858371 0.77 THRB (0.78) THRBTHRAPPARGRXRA
SCHEMBL5859435 0.76 THRB (0.60) THRBTHRAPPARG
SCHEMBL28118607 0.75 GAA (0.52) THRBTHRAPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1862450-A2 Novel compounds KARO BIO AB (SE) 2007-12-05 EP disclosed
EP-1537073-B1 BENZAMIDE OR PHENYLACETAMIDE DERIVATIVES USEFUL AS THYROID RECEPTOR LIGANDS KAROBIO AB (SE) 2007-09-12 EP disclosed
US-7153997-B2 Benzamide derivatives as thyroid receptor ligands KARO BIO AB (SE) 2006-12-26 US disclosed
US-20060135614-A1 Novel compounds NORIN, THOMAS ANDERS WILSON (SE) 2006-06-22 US disclosed
EP-1537073-A2 BENZAMIDE OR PHENYLACETAMIDE DERIVATIVES USEFUL AS THYROID RECEPTOR LIGANDS KARO BIO AB (SE) 2005-06-08 EP disclosed
WO-2004007430-A2 BENZAMIDE OR PHENYLACETAMIDE DERIVATIVES USEFUL AS THYROID RECEPTOR LIGANDS KARO BIO AB (SE) 2004-01-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060135614-A1 Novel compounds THRB, TSHR, THRA THRB 1/4885THRA 3/4885PPARG 14/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.