Gemcabene

Gemcabene

SCHEMBL528316

CC(C)(CCCCOCCCCC(C)(C)C(=O)O)C(=O)O.[CaH2]

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACLY P53396 1/20 0.53
ACACB O00763 1/20 0.52
ACACA Q13085 1/20 0.52
PPARA Q07869 7/20 0.45
TTR P02766 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C8 P10632 1/20 0.42
CHRM1 P11229 1/20 0.42
CYP2C9 P11712 1/20 0.42
TSHR P16473 1/20 0.42
ADRA1A P35348 1/20 0.42
PPARG P37231 1/20 0.42
HTR2B P41595 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
SLCO1B3 Q9NPD5 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
CISD1 Q9NZ45 1/20 0.42
SLCO1B1 Q9Y6L6 1/20 0.42
LTB4R Q15722 4/20 0.42
CYP4F2 P78329 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Gemcabene SCHEMBL4184554 1.00 ACLY (0.53) ACLYACACBACACAPPARATTR
Gemcabene SCHEMBL761631 0.98 ACLY (0.55) ACLYACACBACACAPPARATTR
SCHEMBL14269711 0.96 ACLY (0.59) ACLYACACBACACAPPARATTR
SCHEMBL5524941 0.96 ACLY (0.59) ACLYACACBACACAPPARATTR
SCHEMBL5531453 0.96 ACLY (0.59) ACLYACACBACACAPPARATTR
SCHEMBL6258161 0.96 ACLY (0.53) ACLYACACBACACAPPARATTR
SCHEMBL5521484 0.94 ACLY (0.57) ACLYACACBACACAPPARATTR
SCHEMBL6267270 0.94 ACLY (0.52) ACLYACACBACACAPPARATTR
SCHEMBL13210381 0.92 ACLY (0.50) ACLYACACBACACAPPARATTR
SCHEMBL5528996 0.91 ACLY (0.52) ACLYACACBACACAPPARATTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 34 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1715891-B2 METHODS OF TREATING OSTEOARTHRITIS WITH ANTI-IL-6 ANTIBODIES WARNER LAMBERT CO (US) 2014-08-13 EP claimed
US-20100215654-A1 Methods of treating Osteoarthritis with IL-6 Antagonists PFIZER, INC. (US) 2010-08-26 US claimed
EP-1715891-B1 METHODS OF TREATING OSTEOARTHRITIS WITH ANTI-IL-6 ANTIBODIES WARNER LAMBERT CO (US) 2010-04-21 EP claimed
US-20080145367-A1 Methods of Treating Osteoarthritis with Il-6 Antagonists WARNER-LAMBERT COMPAY, LLC 2008-06-19 US claimed
US-20070203212-A1 METHOD OF TREATING OSTEOARTHRITIS WARNER-LAMBERT COMPANY (US) 2007-08-30 US claimed
EP-1715891-A2 METHODS OF TREATING OSTEOARTHRITIS WITH ANTI-IL-6 OR ANTI-IL6 RECEPTOR ANTIBODIES Warner-Lambert Company LLC (US) 2006-11-02 EP claimed
WO-2005080429-A2 METHODS OF TREATING OSTEOARTHRITIS WITH ANTI-IL-6 OR ANTI-IL6 RECEPTOR ANTIBODIES WARNER-LAMBERT COMPANY LLC (US) 2005-09-01 WO claimed
US-20050148654-A1 Statin-carboxyalkylether combinations BISGAIER CHARLES L (US) 2005-07-07 US claimed
EP-1539127-A1 METHOD OF TREATING OSTEOARTHRITIS WARNER-LAMBERT COMPANY LLC (US) 2005-06-15 EP claimed
US-20040072903-A1 Carboxyalkylether-acat inhibitors combinations AUERBACH BRUCE JEFFREY (US) 2004-04-15 US claimed
US-20040048910-A1 Dialkyl ether di-substituted with formyl, carboxy acid, ester and/or tetrazole, which are on tertiary carbon atoms, e.g., 6-(5-carboxy-5-methylhexyloxy)-2,2-dimethylhexanoic acid; lupus, connective tissue disease, sepsis, joint pain WARNER-LAMBERT COMPANY 2004-03-11 US claimed
WO-2004017952-A1 METHOD OF TREATING OSTEOARTHRITIS WARNER-LAMBERT COMPANY LLC (US) 2004-03-04 WO claimed
EP-1292363-A2 CARBOXYALKYLETHER-ACAT INHIBITOR COMBINATIONS WARNER-LAMBERT COMPANY (US) 2003-03-19 EP claimed
WO-2001093845-A2 CARBOXYALKYLETHER-ACAT INHIBITOR COMBINATIONS WARNER-LAMBERT COMPANY (US) 2001-12-13 WO claimed
US-12503422-B2 Gemcabene, pharmaceutically acceptable salts thereof, compositions thereof and methods of use therefor NEUROBO PHARMACEUTICALS, INC. (US) 2025-12-23 US disclosed
US-20220332672-A1 GEMCABENE, PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF, COMPOSITIONS THEREOF AND METHODS OF USE THEREFOR NEUROBO PHARMACEUTICALS INC (US) 2022-10-20 US disclosed
CN-111704543-A Process and intermediates for preparing alpha, omega-dicarboxylic acid terminated dialkyl ethers 燿石治疗公司 2020-09-25 CN disclosed
US-20040167229-A1 Method of lowering CRP and reducing systemic inflammation BAKKER-ARKEMA REBECCA (US) 2004-08-26 US disclosed
WO-2004045596-A1 METHOD OF LOWERING CRP AND REDUCING SYSTEMIC INFLAMMATION WARNER-LAMBERT COMPANY LLC (US) 2004-06-03 WO disclosed
CN-1395555-A Calcium dicarboxylate ethers, method of making same, and treatment of vascular disease and diabetes therewith WARNER LAMBERT CO (US) 2003-02-05 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220332672-A1 GEMCABENE, PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF, COMPOSITIONS THEREOF AND METHODS OF USE THEREFOR NPC1L1, NOTUM, CEL ACLY 2298/4885ACACB 1237/4885ACACA 1161/4885
US-20040048910-A1 Dialkyl ether di-substituted with formyl, carboxy acid, ester and/or tetrazole, which are on tertiary carbon atoms, e.g., 6-(5-carboxy-5-methylhexyloxy)-2,2-dimethylhexanoic acid; lupus, connective tissue disease, sepsis, joint pain TLR5, SSB, TLR4 ACLY 3034/4885ACACB 2221/4885ACACA 1120/4885
US-20070203212-A1 METHOD OF TREATING OSTEOARTHRITIS SYVN1, MMP13, TNF ACLY 560/4885ACACB 412/4885ACACA 228/4885
US-20050148654-A1 Statin-carboxyalkylether combinations HMGCR, CETP, LCAT ACLY 436/4885ACACB 29/4885ACACA 26/4885
US-12503422-B2 Gemcabene, pharmaceutically acceptable salts thereof, compositions thereof and methods of use therefor NPC1L1, NOTUM, CEL ACLY 2298/4885ACACB 1237/4885ACACA 1161/4885
US-20040072903-A1 Carboxyalkylether-acat inhibitors combinations LCAT, CETP, ACAT2 ACLY 98/4885ACACB 17/4885ACACA 5/4885
US-20040167229-A1 Method of lowering CRP and reducing systemic inflammation ALB, TTR, IL6 ACLY 2661/4885ACACB 1828/4885ACACA 1857/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.