SCHEMBL5288721

SCHEMBL5288721

Cc1ccc(-c2cc(=O)n(CC#N)c(=O)n2-c2ccc([S+](C)[O-])cc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.41
PTGS2 P35354 4/20 0.37
PTGS1 P23219 2/20 0.37
THRB P10828 1/20 0.36
CYP2C9 P11712 1/20 0.34
HTT P42858 1/20 0.34
ALDH1A1 P00352 4/20 0.33
KDM4E B2RXH2 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
CHRNA7 P36544 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
LMNA P02545 1/20 0.33
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5292958 0.83 PTGS2 (0.56) PTGS2PTGS1CYP2C9
SCHEMBL5280436 0.76 POLB (0.37) POLBPTGS2PTGS1THRBCYP2C9
SCHEMBL5294487 0.75 POLB (0.39) POLBPTGS2PTGS1HTTALDH1A1
SCHEMBL14624160 0.71 HTT (0.35) POLBPTGS2PTGS1THRBCYP2C9
SCHEMBL14624155 0.71 KDM4E (0.33) POLBPTGS2PTGS1CYP2C9HTT
SCHEMBL5296183 0.69 POLB (0.34) POLBPTGS2PTGS1THRBCYP2C9
SCHEMBL5325697 0.68 RAD51 (0.40) PTGS2PTGS1THRBCYP2C9HTT
SCHEMBL5331474 0.67 PTGS2 (0.38) PTGS2PTGS1THRBCYP2C9HTT
SCHEMBL14622453 0.67 CYP11B1 (0.43) POLBHTTALDH1A1KDM4EGAA
SCHEMBL5297375 0.65 MEN1 (0.42) POLBPTGS2CYP2C9HTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007007161-A2 NOVEL BIO-ACTIVE DERIVATIVES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-01-18 WO disclosed
WO-2007007161-A2 NOVEL BIO-ACTIVE DERIVATIVES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-01-18 WO disclosed