SCHEMBL14624155

SCHEMBL14624155

CSc1ccc(-c2cc(=O)n(CC#N)c(=O)n2-c2ccc(C(C)(C)C)cc2)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
MDM2 Q00987 1/20 0.33
NPC1 O15118 1/20 0.33
S1PR4 O95977 1/20 0.33
HSP90AA1 P07900 1/20 0.33
MAPT P10636 1/20 0.33
S1PR1 P21453 1/20 0.33
MAPK1 P28482 1/20 0.33
AGTR1 P30556 1/20 0.33
OPRK1 P41145 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
EPHX2 P34913 1/20 0.33
NR1H4 Q96RI1 1/20 0.33
PTGS2 P35354 5/20 0.32
GRIA2 P42262 2/20 0.31
GRIA4 P48058 2/20 0.31
POLB P06746 1/20 0.31
PTGS1 P23219 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5281280 0.87 PTGS2 (0.39) KDM4EPTGS2PTGS1
SCHEMBL5288747 0.85 PTGS2 (0.38) KDM4EALDH1A1NPC1MAPTOPRK1
SCHEMBL5288324 0.84 L3MBTL1 (0.36) KDM4EALDH1A1NPC1MAPTPTGS2
SCHEMBL14624160 0.77 HTT (0.35) NPC1MAPK1HTTSMN1; SMN2PTGS2
SCHEMBL5296183 0.75 POLB (0.34) KDM4EALDH1A1HTTSMN1; SMN2PTGS2
SCHEMBL5325697 0.74 RAD51 (0.40) NPC1MAPK1HTTSMN1; SMN2PTGS2
SCHEMBL5280436 0.73 POLB (0.37) KDM4EALDH1A1MAPTHTTPTGS2
SCHEMBL5331474 0.73 PTGS2 (0.38) KDM4EMAPTHTTSMN1; SMN2PTGS2
SCHEMBL14622453 0.72 CYP11B1 (0.43) KDM4EALDH1A1NPC1MAPK1HTT
SCHEMBL5325289 0.72 HSP90AA1 (0.38) NPC1HSP90AA1MAPTMAPK1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007007161-A2 NOVEL BIO-ACTIVE DERIVATIVES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-01-18 WO disclosed