SCHEMBL5280436

SCHEMBL5280436

CSc1ccc(-n2c(-c3ccc(C)cc3)cc(=O)n(CC#N)c2=O)cc1F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.37
ALDH1A1 P00352 6/20 0.31
KDM4E B2RXH2 3/20 0.31
HPGD P15428 1/20 0.31
PPARG P37231 1/20 0.31
NCOA2 Q15596 1/20 0.31
NCOA1 Q15788 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
NCOA3 Q9Y6Q9 1/20 0.31
PTGS2 P35354 5/20 0.31
PTGS1 P23219 3/20 0.31
TDP1 Q9NUW8 2/20 0.30
MAPT P10636 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
RAD51 Q06609 1/20 0.30
THRB P10828 1/20 0.30
CYP2C9 P11712 1/20 0.30
HTT P42858 1/20 0.30
MEN1 O00255 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5281280 0.79 PTGS2 (0.39) KDM4EPTGS2PTGS1
SCHEMBL5288324 0.78 L3MBTL1 (0.36) POLBALDH1A1KDM4EPTGS2MAPT
SCHEMBL5292958 0.77 PTGS2 (0.56) PTGS2PTGS1CYP2C9
SCHEMBL5288721 0.76 POLB (0.41) POLBALDH1A1KDM4EHPGDNPSR1
SCHEMBL14624160 0.73 HTT (0.35) POLBPTGS2PTGS1RAD51THRB
SCHEMBL14624155 0.73 KDM4E (0.33) POLBALDH1A1KDM4ENPSR1PTGS2
SCHEMBL5294487 0.73 POLB (0.39) POLBALDH1A1KDM4ENPSR1PTGS2
SCHEMBL5296183 0.71 POLB (0.34) POLBALDH1A1KDM4EHPGDPTGS2
SCHEMBL5325697 0.70 RAD51 (0.40) PTGS2PTGS1RAD51THRBCYP2C9
SCHEMBL5331474 0.69 PTGS2 (0.38) KDM4EPTGS2PTGS1MAPTTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007007161-A2 NOVEL BIO-ACTIVE DERIVATIVES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-01-18 WO claimed
WO-2007007161-A2 NOVEL BIO-ACTIVE DERIVATIVES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-01-18 WO disclosed
WO-2007007161-A2 NOVEL BIO-ACTIVE DERIVATIVES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-01-18 WO disclosed