SCHEMBL529294

SCHEMBL529294

Oc1cc(NCCN2CCNCC2)ccc1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.47
HSP90AA1 P07900 2/20 0.47
HSP90AB1 P08238 1/20 0.47
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
CA9 Q16790 2/20 0.44
KHK P50053 1/20 0.43
MELK Q14680 1/20 0.42
CYP2D6 P10635 2/20 0.41
CYP1A2 P05177 1/20 0.41
HTR7 P34969 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
ALDH1A1 P00352 2/20 0.39
HTR4 Q13639 1/20 0.39
KDM4E B2RXH2 2/20 0.39
HSD17B10 Q99714 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
GAA P10253 2/20 0.39
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16477242 0.81 HTR4 (0.46) SIGMAR1HSP90AA1HSP90AB1CA1CA2
SCHEMBL5752131 0.74 SIGMAR1 (0.53) SIGMAR1CA1CA2CA9KHK
SCHEMBL7672095 0.72 SIGMAR1 (0.53) SIGMAR1CA1CA2CA9KHK
SCHEMBL7788377 0.72 CASP6 (0.51) HSP90AA1HSP90AB1CA1CA2CA9
SCHEMBL5159903 0.72 LMNA (0.44) MEN1KMT2AALDH1A1HSD17B10L3MBTL1
SCHEMBL5159107 0.71 IDO1 (0.42) SIGMAR1CYP2D6CYP1A2MEN1KMT2A
SCHEMBL8304884 0.70 CYP3A4 (0.63) SIGMAR1CA1CA2CA9KHK
SCHEMBL9892421 0.70 KHK (0.40) SIGMAR1CA1CA2CA9KHK
SCHEMBL16335399 0.70 ALDH1A1 (0.46) SIGMAR1HSP90AA1HSP90AB1MEN1KMT2A
SCHEMBL453843 0.66 IL1B (0.43) HSP90AA1MEN1KMT2AALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2597955-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME OncoTherapy Science, Inc. (JP) 2013-06-05 EP disclosed
WO-2012016082-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2012-02-02 WO disclosed